871837-60-4
871837-60-4
Chemical Structure
DRAK2-IN-1
- CAS No.: 871837-60-4
- Formula:C21H20N4O3
- Molecular Weight:376.41
IUPAC Name: N-((2Z,3Z)-3-(hydroxyimino)-2'-oxo-[2,3'-biindolinylidene]-5'-yl)pentanamide
InChIKey: QSDUMEKQISKWQM-PMBVCKSESA-N
SMILES: CCCCC(NC1=CC2=C(NC(/C2=C3NC4=C(C=CC=C4)C\3=N\O)=O)C=C1)=O
Biological Activity: DRAK2-IN-1, compound 16, is a potent, selective and ATP-competitive DRAK2 inhibitor with IC50and Kivalues of 3 nM and 0.26 nM, respectively. DRAK2-IN-1 also has inbitory effect on DRAK1 (IC50=51 nM)[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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DRAK2-IN-1 | 99.93% | DRAK2-IN-1, compound 16, is a potent, selective and ATP-competitive DRAK2 inhibitor with IC50and Kivalues of 3 nM and 0.26 nM, respectively. DRAK2-IN-1 also has inbitory effect on DRAK1 (IC50=51 nM). | ||||||||||||||||||||
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References
Keywords
