1. Apoptosis
  2. DAPK
  3. DRAK2-IN-1

DRAK2-IN-1 

Cat. No.: HY-122629
Handling Instructions

DRAK2-IN-1, compound 16, is a potent, selective and ATP-competitive DRAK2 inhibitor with IC50and Kivalues of 3 nM and 0.26 nM, respectively. DRAK2-IN-1 also has inbitory effect on DRAK1 (IC50=51 nM).

For research use only. We do not sell to patients.

DRAK2-IN-1 Chemical Structure

DRAK2-IN-1 Chemical Structure

CAS No. : 871837-60-4

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Description

DRAK2-IN-1, compound 16, is a potent, selective and ATP-competitive DRAK2 inhibitor with IC50and Kivalues of 3 nM and 0.26 nM, respectively. DRAK2-IN-1 also has inbitory effect on DRAK1 (IC50=51 nM)[1].

IC50 & Target

IC50: 3 nM (DRAK2); 51 nM (DRAK1); 1.8 μM (DRPK2); 2.3 μM (DRAK2); 1.8 μM (DRPK3)[1]

Molecular Weight

376.41

Formula

C₂₁H₂₀N₄O₃

CAS No.

871837-60-4

SMILES

CCCCC(NC1=CC2=C(NC(/C2=C3NC4=C(C=CC=C4)C\3=N\O)=O)C=C1)=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
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Keywords:

DRAK2-IN-1DAPKDeath associated protein kinaseInhibitorinhibitorinhibit

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