93361-66-1
Chemical Structure
Histargin
- CAS No.: 93361-66-1
- Formula:C14H25N7O4
- Molecular Weight:355.39
IUPAC Name: (2-(((S)-1-carboxy-2-(1H-imidazol-5-yl)ethyl)amino)ethyl)-L-arginine
InChIKey: LLPMPMKLOHAIMY-QWRGUYRKSA-N
SMILES: N=C(N)NCCC[C@@H](C(O)=O)NCCN[C@H](C(O)=O)CC1=CN=CN1
Biological Activity: Histargin is a selective carboxypeptidase B inhibitor with an IC50 of 17 μg/mL and a Ki of 30 μM. Histargin exerts competitive inhibition with substrate, with inhibitory activity abolished by metal cations. Histargin shows no significant inhibitory activity against carboxypeptidase A, aminopeptidase A, or aminopeptidase B[1].
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Histargin | Histargin is a selective carboxypeptidase B inhibitor with an IC50 of 17 μg/mL and a Ki of 30 μM. Histargin exerts competitive inhibition with substrate, with inhibitory activity abolished by metal cations. Histargin shows no significant inhibitory activity against carboxypeptidase A, aminopeptidase A, or aminopeptidase B. | |||||||||||||||||||||
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Keywords
