CysLT1/2 receptor antagonist-1
CysLT1/2 receptor antagonist-1 is a dual CysLT1 and CysLT2 receptor antagonist with IC50 values of 0.044 μM (CysLT1) and 0.17 μM (CysLT2). CysLT1/2 receptor antagonist-1 can be used for the research of bronchial asthma.
For research use only. We do not sell to patients.
- CAS No.: 1637756-67-2
- Formula: C31H34N2O7
- Molecular Weight:546.61
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All Leukotriene Receptor Isoforms
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Biological Activity
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CysLT1 0.044 μM (IC50) |
CysLT2 0.17 μM (IC50) |
CysLT1/2 receptor antagonist-1 (Compound 11b) antagonizes CysLT1 and CysLT2 receptors, with an IC50 value of 0.044 μM against CysLT1 and 0.17 μM against CysLT2[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 1637756-67-2
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Molecular Weight 546.61
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Formula C31H34N2O7
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SMILES
O=C(CCCCN1C2=C(OC(C1)C(O)=O)C(NC(C3=CC=C(C=C3)OCCCCC4=CC=CC=C4)=O)=CC=C2)O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)