1. Signaling Pathways
  2. GPCR/G Protein
  3. Leukotriene Receptor
  4. LTD4/CysLT1 Inhibitors

LTD4/CysLT1 Inhibitors

LTB4

LTC4

LTD4/CysLT1

LTE4

CysLT2

CysLT1

Your Search Returned No Results.

Sorry. There is currently no product that acts on isoform LTD4/CysLT1 together.

Please try each isoform separately.

LTD4/CysLT1 Specific Antagonists
Product Name LTD4/CysLT1 LTC4 LTE4 LTD4/CysLT1 Selectivity Purity
MK-571 sodium salt
LTD4, Ki: 0.22 nM (In guinea pig lung)
LTD4, Ki: 2.1 nM (In human lung)
    Selective Antagonist 99.24%
Montelukast sodium
CysLT1
    Selective Antagonist 99.82%
Zafirlukast
LTD4
    Selective Antagonist 99.10%
CP-96486
LTD4, Ki: 20 nM
    Selective Antagonist
Iralukast
CysLT1, pKi: 7.8
    Selective
RS-601
LTD4
    Selective Antagonist
LTD4 antagonist 1
LTD4, Ki: 0.57 nM
    Selective Antagonist
KP496
LTD4
    Selective Antagonist
YM158 free base
LTD4, pA2: 8.87
    Selective Antagonist
Pranlukast hemihydrate
LTD4, Ki: 0.99 nM
LTC4, Ki: 5640 nM
LTE4, Ki: 0.63 nM
Pan Antagonist 99.93%
LM-1484
CysLT1
LTC4
  Pan Antagonist
Tipelukast
LTD4, pA2: 6.41 (In guinea-pigs)
 
LTE4, pA2: 6.45 (In guinea-pigs)
Pan Antagonist