Ghrelin receptor full agonist-2
Ghrelin receptor full agonist-2 (compound 12j) is a highly potent Ghrelin receptor full agonist.
For research use only. We do not sell to patients.
- CAS No.: 2602452-73-1
- Formula: C26H28ClN5O5S
- Molecular Weight:558.05
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| HEK293 | EC50 |
0.442 nM
Compound: 12j
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Agonist activity at human GHSR expressed in HEK293 cells assessed as increase in IP1 accumulation measured after 90 mins in presence of LiCl by HTRF assay
Agonist activity at human GHSR expressed in HEK293 cells assessed as increase in IP1 accumulation measured after 90 mins in presence of LiCl by HTRF assay
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[PMID: 32787075] |
| HEK293 | EC50 |
0.9 nM
Compound: 12j
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Agonist activity at dog GHSR expressed in HEK293 cells assessed as increase in IP1 accumulation measured after 60 mins in presence of LiCl by HTRF assay
Agonist activity at dog GHSR expressed in HEK293 cells assessed as increase in IP1 accumulation measured after 60 mins in presence of LiCl by HTRF assay
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[PMID: 32787075] |
Chemical Information
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CAS No. 2602452-73-1
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Molecular Weight 558.05
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Formula C26H28ClN5O5S
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SMILES
O=C(C1=NOC(C2=C(C=CC=C2)Cl)=C1)N[C@@H]3[C@H](CN(C3)S(=O)(C4=CC=CC=C4)=O)C(N[C@H]5CCCNC5)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Ghrelin receptor full agonist-2 Related Classifications
HY-145364 Related Classifications
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