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Cat. No.: HY-P0036S

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Octreotide-d₈ TFA

(Synonyms: SMS 201-995-d8 TFA)

Octreotide-d₈ (SMS 201-995-d₈) TFA is the deuterium labeled Octreotide TFA. Octreotide (SMS 201-995) is a somatostatin receptor agonist and synthetic octapeptide endogenous somatostatin analogue. Octreotide (SMS 201-995) can bind to the somatostatin receptor and mainly subtypes 2, 3, and 5, increases Gi activity, and reduces intracellular cAMP production. Octreotide (SMS 201-995) has antitumor activity, mediates apoptosis and may also be used in disease studies in acromegaly.

For research use only. We do not sell to patients.

Formula: C₅₃H₆₀D₈F₆N₁₀O₁₄S₂
Molecular Weight:1255.34

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Octreotide-d₈ TFA Chemical Structure

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Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- Description
- In Vitro
- Application
Chemical Information
Purity & Documentation
Calculators
Help & FAQs
Classifications
Bioz

Biological Activity

Description

All Somatostatin Receptor Isoforms :

In Vitro

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs.

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Application

1. This compound can be used as a tracer
2. This compound can be used as an internal standard for quantitative analysis by NMR, GC-MS, or LC-MS.

Chemical Information

Molecular Weight 1255.34
Formula C₅₃H₆₀D₈F₆N₁₀O₁₄S₂
SMILES

OC(C(F)(F)F)=O.OC(C(F)(F)F)=O.[2H][C@@](C([2H])(C(C([2H])=C(C([2H])=C1[2H])[2H])=C1[2H])[2H])(C(N[C@H](C(N[C@H](C(N[C@@H]2CC3=CNC4=CC=CC=C43)=O)CC5=CC=CC=C5)=O)CSSC[C@@H](C(N[C@@H]([C@@H](C)O)CO)=O)NC([C@@](NC([C@H](CCCCN)NC2=O)=O)([C@@H](C)O)[H])=O)=O)N
Synonyms

SMS 201-995-d8 TFA
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.