Protein kinase inhibitor 5
Protein kinase inhibitor 5 is a potent TRK-A inhibitor with an IC50 value of 1.8 nM. Protein kinase inhibitor 5 inhibits cell viability.
For research use only. We do not sell to patients.
- CAS No.: 2278204-94-5
- Formula: C29H31F2N7O
- Molecular Weight:531.60
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
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TrkA 1.8 nM (IC50) |
Protein kinase inhibitor 5 (compound 2) (0.014-10 µM; 72 h) inhibits cell viability with a GI50 value of <1 nM for TEL-NTRK1-BaF3 cells[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 2278204-94-5
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Molecular Weight 531.60
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Formula C29H31F2N7O
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SMILES
O=C(NC1=C2N=C(N3[C@@H](C4=CC(F)=CC=C4F)CCC3)C=CN2N=C1)C5=CC=C(CN6CCN(C)CC6)C=C5
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Protein kinase inhibitor 5 Related Classifications
HY-153745 Related Classifications
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