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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
3 Results for "
(R)-Baclofen
" in MedChemExpress (MCE) Product Catalog:
Products (3)
3 Results for "(R)-Baclofen" in MCE Product Catalog:
2
Target:
Research Areas:
(R)-Baclofen (Arbaclofen) is a selective GABAB receptor agonist .
2
2 Cited Publications
Cat. No.: HY-17354A
CAS No.: 63701-55-3
Synonyms: ArBaclofen hydrochloride; STX 209 hydrochloride
Target:
Research Areas:
(R)-Baclofen hydrochloride (Arbaclofen hydrochloride) is a selective GABAB receptor agonist .
Cat. No.: HY-114076
CAS No.: 150175-54-5
Target:
Research Areas:
CGP55845 is a potent and selective GABAB receptor antagonist with activity that blocks agonist binding. The IC50 value of CGP55845 is 5 nM, indicating that it exhibits significant activity in inhibiting GABA and glutamate release. The apparent Kd of CGP55845 when forming a complex with the GABAB receptor is 30 nM, indicating its high affinity for this receptor. CGP55845 is as potent as 100 μM CGP 35348 in relieving the inhibitory effect of (R)-(-)-baclofen .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
