1 Result for "

2387510-80-5

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "2387510-80-5" in MCE Product Catalog:

2
2 Cited Publications
Cat. No.: HY-114209
CAS No.: 2387510-80-5
Purity:  99.84%
Research Areas:  

Cancer

MRK-740, a chemical probe, is a potent, selective and substrate-competitive PRDM9 histone methyltransferase inhibitor with an IC50 of 80?nM. MRK-740 is more selective for PRDM9 than other histone methyltransferases and other non-epigenetic targets. MRK-740 reduces PRDM9-dependent trimethylation of H3K4 (IC50?=?0.8?μM) .
loading...
    loading...