1 Result for "

2953426-48-5

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "2953426-48-5" in MCE Product Catalog:

Cat. No.: HY-143905
CAS No.: 2953426-48-5
Target:  

PROTACs Mps1

Research Areas:  

Cancer

PROTAC TTK degrader-2 is a threonine tyrosine kinase (TTK) PROTAC degrader with a DC50 of 3.1 nM in COLO-205 cells. PROTAC TTK degrader-2 induces proteasome-mediated degradation of TTK. It inhibits the proliferation of colorectal cancer cells. In colorectal cancer xenograft mouse models, PROTAC TTK degrader-2 mediates target degradation and exerts anticancer activity. PROTAC TTK degrader-2 can be used in colorectal cancer-related research .
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