3 Results for "

5-Hydroxymethyl tolterodine formate

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "5-Hydroxymethyl tolterodine formate" in MCE Product Catalog:

Cat. No.: HY-76569B
CAS No.: 380636-49-7
Synonyms: PNU-200577 formic
Target:  

mAChR

Research Areas:  

Neurological Disease

5-Hydroxymethyl tolterodine (formate) (PNU-200577 (formic)) is an active metabolite of the muscarinic acetylcholine receptor antagonists Tolterodine (HY-A0024) and Fesoterodine (HY-70053). 5-Hydroxymethyl tolterodine (formate) is formed from tolterodine by the cytochrome P450 (CYP) isoform CYP2D6 and from fesoterodine by plasma esterases.
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Cat. No.: HY-76570S1
5-Hydroxymethyl Tolterodine-d14 (formate) is deuterium labeled (Rac)-5-Hydroxymethyl Tolterodine. (Rac)-5-Hydroxymethyl Tolterodine ((Rac)-Desfesoterodine), an active metabolite of Tolterodine, is a mAChR antagonist (Ki values of 2.3 nM, 2 nM, 2.5 nM, 2.8 nM, and 2.9 nM for M1, M2, M3, M4, and M5 receptors, respectively). (Rac)-5-Hydroxymethyl Tolterodine can be used for overactive bladder research .
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Cat. No.: HY-76996S1
(S)-5-Hydroxymethyl Tolterodine-d14 (formate) is deuterium labeled (S)-2-(3-(diisopropylamino)-1-phenylpropyl)-4-(hydroxymethyl)phenol.
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