3 Results for "

866021-03-6

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "866021-03-6" in MCE Product Catalog:

Cat. No.: HY-14325A
CAS No.: 866021-03-6
Target:  

Dopamine Receptor

Research Areas:  

Neurological Disease

L-745870 trihydrochloride is a potent, selective, brain-penetrant and orally active dopamine D4 receptor antagonist with a Ki of 0.43 nM. L-745870 trihydrochloride shows weaker affinity for D2 (Ki of 960 nM) and D3 (Ki of 2300 nM) receptors, and exhibits moderate affinity for 5-HT2 receptors, sigma sites and α-adrenoceptors .
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3
3 Cited Publications
Cat. No.: HY-14325
CAS No.: 158985-00-3
Purity:  99.50%
Target:  

Dopamine Receptor

Research Areas:  

Neurological Disease

L-745870 is a potent, selective, brain-penetrant and orally active dopamine D4 receptor antagonist with a Ki of 0.43 nM. L-745870 shows weaker affinity for D2 (Ki of 960 nM) and D3 (Ki of 2300 nM) receptors, and exhibits moderate affinity for 5-HT2 receptors, sigma sites and α-adrenoceptors .
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3
3 Cited Publications
Cat. No.: HY-14325B
CAS No.: 1173023-36-3
Purity:  99.91%
Target:  

Dopamine Receptor

Research Areas:  

Neurological Disease

L-745870 hydrochloride is a potent, selective, brain-penetrant and orally active dopamine D4 receptor antagonist with a Ki of 0.43 nM. L-745870 hydrochloride shows weaker affinity for D2 (Ki of 960 nM) and D3 (Ki of 2300 nM) receptors, and exhibits moderate affinity for 5-HT2 receptors, sigma sites and α-adrenoceptors .
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