1 Result for "

AXL/Angiokinase-IN-1

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "AXL/Angiokinase-IN-1" in MCE Product Catalog:

Cat. No.: HY-170776
Target:  

PDGFR VEGFR FGFR Apoptosis

Research Areas:  

Cancer

AXL/Angiokinase-IN-1 (compound 11b) is an AXL/triple angiokinase inhibitor, IC50=3.75 nM (AXL expression). AXL/Angiokinase-IN-1 inhibits epithelial-mesenchymal transition (EMT) in Bxpc-3, blocking lung cancer cell metastasis. AXL/Angiokinase-IN-1 also inhibits vascular and fibroblast functions, promoting apoptosis (apoptosis) in cancer cells and fibroblasts. AXL/Angiokinase-IN-1 features low toxicity and good metabolic stability .
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