2 Results for "

Afimoxifene (Standard)

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "Afimoxifene (Standard)" in MCE Product Catalog:

(E/Z)-4-Hydroxytamoxifen (Standard)
(E/Z)-4-Hydroxytamoxifen (Standard)
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Cat. No.: HY-16950AR
CAS No.: 68392-35-8
Synonyms: Afimoxifene (Standard); 4-OHT (Standard)
Category:  

Alkaloids Monophenols Other Alkaloids Phenols Endogenous metabolite

Target:  

Reference Standards Estrogen Receptor/ERR Endogenous Metabolite

(E/Z)-4-Hydroxytamoxifen (Standard) is the analytical standard of (E/Z)-4-Hydroxytamoxifen. This product is intended for research and analytical applications. (E/Z)-4-Hydroxytamoxifen (Afimoxifene) is a racemic compound of (Z)-4-Hydroxytamoxifen and (E)-4-Hydroxytamoxifen isomers. (E/Z)-4-Hydroxytamoxifen is a selective estrogen receptor modulator with mixed estrogenic and antiestrogenic activity, which is also an active metabolite of Tamoxifen (HY-13757A). (E/Z)-4-Hydroxytamoxifen is an agonist of the G protein-coupled estrogen receptor (GPER) with relatively low affinity (100-1000 nM). (E/Z)-4-Hydroxytamoxifen is promising for research of cyclical mastalgia, such as breast pain, tenderness, and nodularity .
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4-Hydroxytamoxifen (Standard)
4-Hydroxytamoxifen (Standard)
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Cat. No.: HY-16950R
CAS No.: 68047-06-3
Synonyms: (Z)-4-Hydroxytamoxifen (Standard); trans-4-Hydroxytamoxifen (Standard); (Z)-Afimoxifene (Standard)
Target:  

Estrogen Receptor/ERR Reference Standards

Research Areas:  

Cancer

4-Hydroxytamoxifen (Standard) is the analytical standard of 4-Hydroxytamoxifen. This product is intended for research and analytical applications. 4-Hydroxytamoxifen ((Z)-4-Hydroxytamoxifen) is an orally active, selective estrogen receptor modulator (SERM). 4-Hydroxytamoxifen ((Z)-4-Hydroxytamoxifen) is also the active metabolic form of Tamoxifen (HY-13757A) in vivo and can be used to induce gene knockout in transgenic mice expressing CreER .
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