1 Result for "

N-Pentanoyl 2-benzyltryptamine

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "N-Pentanoyl 2-benzyltryptamine" in MCE Product Catalog:

Cat. No.: HY-107628
CAS No.: 220339-00-4
Target:  

Melatonin Receptor

Research Areas:  

Neurological Disease

N-Pentanoyl 2-benzyltryptamine is a potent and selective antagonist of MT2 melatonin receptor, with a pKi of 8.03 for human MT2. N-Pentanoyl 2-benzyltryptamine shows 89- and 229-fold selectivity for human MT2 over human mt1 and Xenopus mel1c receptor subtypes. N-Pentanoyl 2-benzyltryptamine can inhibit melatonin-induced enhancement of electrically-evoked responses .
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