1 Result for "

NMDAR/HDAC-IN-1

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "NMDAR/HDAC-IN-1" in MCE Product Catalog:

Cat. No.: HY-147873
Target:  

iGluR HDAC

Research Areas:  

Neurological Disease

NMDAR/HDAC-IN-1 (Compound 9d) is a dual NMDAR and HDAC inhibitor with a Ki of 0.59 μM for NMDAR and IC50 values of 2.67, 8.00, 2.21, 0.18 and 0.62 μM for HDAC1, HDAC2, HDAC3, HDAC6 and HDAC8, respectively. NMDAR/HDAC-IN-1 efficiently penetrates the blood brain barrier .
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