![[D-Ala2]leucine-enkephalin](https://file.medchemexpress.com/product_pic/hy-p0098.gif "Click to View [D-Ala2]leucine-enkephalin Product Detail")
![[DPen2, Pen5] Enkephalin](https://file.medchemexpress.com/product_pic/hy-p3546.gif "Click to View [DPen2, Pen5] Enkephalin Product Detail")
Scientific Reviews
Product Guides
Blogs
Topics
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
15 Results for "
Opioid analog
" in MedChemExpress (MCE) Product Catalog:
Products (15)
15 Results for "Opioid analog" in MCE Product Catalog:
Cat. No.: HY-P0098
CAS No.: 64963-01-5
Target:
Research Areas:
Cat. No.: HY-W048697
CAS No.: 201532-01-6
Target:
Research Areas:
Cat. No.: HY-P3546
CAS No.: 88373-72-2
Target:
Research Areas:
Cat. No.: HY-174422
CAS No.: 676494-79-4
Target:
Research Areas:
Opioid receptor antagonist 2 (Compound 9) is a potent opioid receptor antagonist. Opioid receptor antagonist 2 can reverse ventilatory depression and vocal cord closure induced by sedative agent analogs in mice. Opioid receptor antagonist 2 is promising for research of acute poisoning such as respiratory depression caused by overdose of opioids .
Cat. No.: HY-172637
CAS No.: 2712312-12-2
Target:
Research Areas:
Phenethyl 4-ANPP is a MOR (μ-opioid receptor) agonist. Phenethyl 4-ANPP is an analytical reference standard that is structurally similar to known opioids .
Target:
Research Areas:
Chlorphine is a neuroactive halogenated opioid analog .
Cat. No.: HY-P3223A
Target:
Research Areas:
Cat. No.: HY-P2199
CAS No.: 137415-20-4
Target:
Research Areas:
Cat. No.: HY-P1577
CAS No.: 115814-08-9
Target:
Research Areas:
Cat. No.: HY-129237
CAS No.: 76995-89-6
Target:
Research Areas:
Azo-enkephalin is an endorphin analog with significant analgesic activity. Azo-enkephalin can be used in the development of opioid analgesics .
Cat. No.: HY-P3223
CAS No.: 126872-95-5
Target:
Research Areas:
Cat. No.: HY-W714509
CAS No.: 41805-63-4
Target:
Research Areas:
AH 8507 structurally belongs to the opioid compounds and is an analog of AH 7563 (HY-W714505). However, AH 8507 does not exhibit significant analgesic effects in mice in both the phenylquinone test and the hot plate test, with ED50 values greater than 100 mg/kg .
Cat. No.: HY-P4679
CAS No.: 103613-84-9
Synonyms: E2078
Target:
Research Areas:
Cat. No.: HY-138232
CAS No.: 141365-20-0
Synonyms: LTNAM
Target:
Research Areas:
Lys-psi(CH2NH)-Trp(Nps)-OMe is a lysine-tryptophan (Nps) pseudodipeptide analog. It is obtained by replacing the peptide bond in the Lys-Trp(Nps) molecule with an aminomethylene bond and has analgesic activity. Lys-psi(CH2NH)-Trp(Nps)-OMe induces a dose-dependent and naloxone-reversible analgesia after intracerebroventricular administration in mice, and its analgesic effect lasts longer than that of the original compound. It protects methionine enkephalin from degradation in rat striatal slices and binds to low-dose opioid peptides to produce analgesia. Lys-psi(CH2NH)-Trp(Nps)-OMe effectively inhibits brain aminopeptidase activity both in vitro and in vivo. The enhanced resistance of this pseudodipeptide to proteolysis may explain its prolonged analgesic activity.
Cat. No.: HY-W241255
CAS No.: 27473-62-7
Research Areas:
Neurological Disease Inflammation/Immunology Endocrinology Cancer
2-Aminoindan-2-carboxylic acid is a conformationally restricted Phenylalanine analog and molecular building block. 2-Aminoindan-2-carboxylic acid constitutes a component of allosteric LFA-1 antagonists targeting the LFA-1/ICAM-1 interaction. 2-Aminoindan-2-carboxylic acid serves as a molecular building block for various biologically active peptides, including μ-receptor-selective opioid analogs, activated protein C inhibitors, and histone deacetylase inhibitors. 2-Aminoindan-2-carboxylic acid can be used in the research of autoimmune diseases, inflammatory diseases, opioid receptor-related diseases, antidiuresis-related diseases, and cancers .
- 1
-
-
Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
