Biphalin acetate
Based on 1 Customer Validation
Biphalin acetate, a BBB-penetrable opioid peptide analog, contains two active enkephalin pharmacophores.Biphalin acetate has high affinity for opioid receptors. Biphalin acetate shows analgesic effect in acute, neuropathic, and chronic animal pain models. Biphalin acetate is also an antiviral, antiproliferative, anti-inflammatory, and neuroprotective agent.
For research use only. We do not sell to patients.
- Formula: C46H56N10O10·xC2H4O2
- Molecular Weight:909.00 (free base)
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Storage:
Sealed storage, away from moisture.
Powder -80°C, 2 years , -20°C, 1 year* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
All Opioid Receptor Isoforms
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Biological Activity
Chemical Information
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Appearance Solid
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Molecular Weight 909.00 (free base)
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Formula C46H56N10O10·xC2H4O2
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Sequence
Tyr-{dAla}-Gly-Phe-NH2 (covalent bridge:Phe-Phe, dimer)
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Sequence Shortening
Y-{D-Ala}-GF-NH2 (covalent bridge:Phe-Phe, dimer)
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Sealed storage, away from moisture
Powder -80°C 2 years -20°C 1 year * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
Purity & Documentation
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Data Sheet (266 KB)
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SDS (252 KB)
- Français - FR (252 KB)
- Deutsch - DE (252 KB)
- Norwegian - NO (252 KB)
- Español - ES (252 KB)
- Swedish - SV (252 KB)
- Italian - IT (252 KB)
- Korean - KR (252 KB)
- Portuguese - PT (252 KB)
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Handling Instructions (2659 KB)
References
[1]. T J Abbruscato, et al. Blood-to-central nervous system entry and stability of biphalin, a unique double-enkephalin analog, and its halogenated derivatives. J Pharmacol Exp Ther. 1996, 276,3. [Content Brief]
[2]. Redkiewicz P, et al. Biphalin-A Potent Opioid Agonist-As a Panacea for Opioid System-Dependent Pathophysiological Diseases? Int J Mol Sci. 2021 Oct 21;22(21):11347. [Content Brief]
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)