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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
9 Results for "
Pitolisant
" in MedChemExpress (MCE) Product Catalog:
Products (9)
9 Results for "Pitolisant" in MCE Product Catalog:
2
2 Cited Publications
Synonyms: Ciproxidine; BF 2649
Target:
Pitolisant hydrochloride is a potent and selective nonimidazole inverse agonist at the recombinant human histamine H3 receptor (Ki=0.16 nM).
2
Target:
Pitolisant is a potent and selective nonimidazole inverse agonist at the recombinant human histamine H3 receptor (Ki=0.16 nM).
Cat. No.: HY-12199A
CAS No.: 362665-57-4
Synonyms: Tiprolisant oxalate
Target:
Pitolisant oxalate is a potent and selective nonimidazole inverse agonist at the recombinant human histamine H3 receptor (Ki=0.16 nM).
Cat. No.: HY-12199R
CAS No.: 362665-56-3
Synonyms: Tiprolisant (Standard)
Pitolisant (Standard) is the analytical standard of Pitolisant. This product is intended for research and analytical applications. Pitolisant is a potent and selective nonimidazole inverse agonist at the recombinant human histamine H3 receptor (Ki=0.16 nM).
Cat. No.: HY-12199S1
CAS No.: 2416991-77-8
Synonyms: Tiprolisant-d6
Cat. No.: HY-12199BR
CAS No.: 903576-44-3
Synonyms: Ciproxidine (Standard); BF 2649 (Standard)
Pitolisant (hydrochloride) (Standard) is the analytical standard of Pitolisant (hydrochloride). This product is intended for research and analytical applications. Pitolisant hydrochloride is a potent and selective nonimidazole inverse agonist at the recombinant human histamine H3 receptor (Ki=0.16 nM).
Cat. No.: HY-12199BS
CAS No.: 2740634-42-6
Synonyms: Ciproxidine-d5 hydrochloride; BF 2649-d5 hydrochloride
Cat. No.: HY-121364
CAS No.: 1416130-06-7
Target:
연구분야:
Bodilisant is a histamine H3 receptor (hH3R) ligand and imaging/labeling agent, with a Ki value of 6.51 nM for hH3R. Bodilisant binds to hH3R to produce strong green fluorescence, localizes to the extracellular membrane without internalization, and generates clear, displaceable fluorescent labeling of hH3R in native human brain tissues. Bodilisant serves as a pharmacological tool to visualize the distribution of hH3R via fluorescence confocal laser scanning microscopy .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
