10 Results for "

Procainamide-d4

" in MedChemExpress (MCE) Product Catalog:
Products (10)

10 Results for "Procainamide-d4" in MCE Product Catalog:

1
1 Cited Publications
Art. -Nr.: HY-P1103
CAS. Nr.: 1030384-98-5
Target:  

CXCR

Forschungsgebiete:  

Cancer

CTCE-9908 is a potent and selective CXCR4 antagonist. CTCE-9908 induces mitotic catastrophe, cytotoxicity and inhibits migration in CXCR4-expressing ovarian cancer cells .
loading...
    loading...
Art. -Nr.: HY-P4070
CAS. Nr.: 1188379-43-2
Target:  

Insulin Receptor

Forschungsgebiete:  

Metabolic Disease

Insulin icodec is an Insulin (HY-P0035) analog that strongly but reversibly binds to albumin. Insulin icodec has long plasma half-life. Insulin icodec modulates insulin receptor activity, controls blood glucose levels, reduces HbA1c levels, and binds reversibly to human serum albumin. Insulin icodec can be used for the research of type 2 diabetes mellitus .
loading...
    loading...
Art. -Nr.: HY-A0084S
Synonyms: Procaine amide-d4 hydrochloride; SP 100-d4 hydrochloride
Procainamide-d4 hydrochloride is deuterated labeled Procainamide. Procainamide hydrochloride is an antiarrhythmic agent used in the study of cardiac arrhythmias.
loading...
    loading...
Art. -Nr.: HY-A0084AS
Synonyms: Procaine amide-d4; SP 100-d4
Procainamide-d4 (Procaine amide-d4) is the deuterium labeled Procainamide (HY-A0084A). Procainamide (Procaine amide) is a specific and potent inhibitor of DNA methyltransferase 1 (DNMT1), which reactivates the expression of tumor suppressor factors by demethylating tumor suppressor genes. Procainamide induces vacuolization in various cell types and reduces cell proliferation and migration. Procainamide relaxes airway smooth muscle by activating potassium channels. Procainamide can be used in cancer and arrhythmia research [4] .
loading...
    loading...
Art. -Nr.: HY-P1103A
Target:  

CXCR

Forschungsgebiete:  

Cancer

CTCE-9908 TFA is a potent and selective CXCR4 antagonist. CTCE-9908 TFA induces mitotic catastrophe, cytotoxicity and inhibits migration in CXCR4-expressing ovarian cancer cells .
loading...
    loading...
Art. -Nr.: HY-P11293
CAS. Nr.: 1309855-53-5
Target:  

Melanocortin Receptor

Forschungsgebiete:  

Cancer

DOTA-GGNle-CycMSHhex is a melanocortin-1 receptor (MC1R)-targeting peptide that can be radionuclide-labeled for melanoma imaging .
loading...
    loading...
Art. -Nr.: HY-P4757
CAS. Nr.: 108081-77-2
Target:  

Parasite

Forschungsgebiete:  

Others

N1-Glutathionyl-spermidine disulfide is a substrate of trypanothione reductase .
loading...
    loading...
Art. -Nr.: HY-P1321
CAS. Nr.: 158859-98-4
Synonyms: 1229U91; GW1229
Forschungsgebiete:  

Neurological Disease

GR231118, an analogue of the C-terminus of neuropeptide Y, is a potent , competitive and relative seletive antagonist at human neuropeptide Y Y receptor with a pKi of 10.4. GR231118 a potent agonist at the human neuropeptide Y Y4 receptor (pEC50=8.6; pKi=9.6) and a weak agonist at the human and rat neuropeptide YY2 and Y5 receptors. GR231118 also has high affinity for the mouse neuropeptide Y Y6 receptor (pKi= 8.8) .
loading...
    loading...
Art. -Nr.: HY-P1321A
Synonyms: 1229U91 TFA; GW1229 TFA
Forschungsgebiete:  

Neurological Disease

GR231118 TFA, an analogue of the C-terminus of neuropeptide Y, is a potent , competitive and relative seletive antagonist at human neuropeptide YY receptor with a pKi of 10.4. GR231118 a potent agonist at the human neuropeptide YY4 receptor (pEC50=8.6; pKi=9.6) and a weak agonist at the human and rat neuropeptide Y Y2 and Y5 receptors. GR231118 also has high affinity for the mouse neuropeptide YY6 receptor (pKi= 8.8) .
loading...
    loading...
Art. -Nr.: HY-P11480
CAS. Nr.: 3105660-96-3
Target:  

Trk Receptor

Forschungsgebiete:  

Neurological Disease

TrkA/NGF-IN-1 (Peptide 19) is an inhibitor of protein-protein interactions between TrkA and NGF (IC50: 21 nM for human TrkA in PathHunter assay). TrkA/NGF-IN-1 shows an analgesic effect in a rat incisional pain model .
loading...
    loading...