2 Results for "

SUCNR1 antagonist-1

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "SUCNR1 antagonist-1" in MCE Product Catalog:

Cat. No.: HY-183639
Research Areas:  

Cancer

SUCNR1 antagonist-1 is an orally active SUCNR1 antagonist. SUCNR1 antagonist-1 forms stable, water-bridged hydrogen bonds with key residue Glu22 1.31 to stabilize binding conformation and modulates protein conformational flexibility. SUCNR1 antagonist-1 blocks succinate-mediated SUCNR1 signaling and induces cell apoptosis. SUCNR1 antagonist-1 can be used for the research of colorectal carcinoma [1].
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1
1 Cited Publications
Cat. No.: HY-150205
CAS No.: 2361972-29-2
Purity:  99.46%
Target:  

Succinate Receptor 1

Research Areas:  

Inflammation/Immunology

Succinate/succinate receptor antagonist 1 is an antagonist of the succinate/succinate receptor. Succinate/succinate receptor antagonist 1 can inhibit the activation of succinate receptor 1 (SUCNR1). Succinate/succinate receptor antagonist 1 can block succinate signaling. Succinate/succinate receptor antagonist 1 can be used for the study of periodontal disease [1].
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