38 Results for "

diketopiperazine

" in MedChemExpress (MCE) Product Catalog:
Products (38)

38 Results for "diketopiperazine" in MCE Product Catalog:

Cat. No.: HY-142104
CAS No.: 934816-82-7
Synonyms: 2-Chlorotrityl Chloride Resin (100-200 mesh,1% DVB,0.4-3.0mmol/g)
Target:  

Drug Intermediate

Research Areas:  

Cancer

2-CTC Resin (100-200 mesh,1% DVB,0.4-3.0mmol/g) is a solid-phase synthesis carrier that has been used to study metabolic disorders in prostate cancer cells. 2-CTC Resin (100-200 mesh,1% DVB,0.4-3.0mmol/g) can be used as a reaction solution of terminal residues and adenine nucleotides to form cyclic peptides. 2-CTC Resin (100-200 mesh,1% DVB,0.4-3.0mmol/g) can prevent racemization during the incorporation of the first protected amino acid and minimized diketopiperazine formation. 2-CTC Resin (100-200 mesh,1% DVB,0.4-3.0mmol/g) is one of the most commonly used and versatile resins available for large-scale production of peptides .
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Cat. No.: HY-101402
CAS No.: 53109-32-3
Synonyms: Cyclohistidyl-proline; Histidylproline diketopiperazine
Cyclo(his-pro) (Cyclo(histidyl-proline)) is an orally active cyclic dipeptide structurally related to tyreotropin-releasing hormone . Cyclo(his-pro) could inhibit NF-κB nuclear accumulation. Cyclo(his-pro) can cross the brain-blood-barrier and affect diverse inflammatory and stress responses .
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Cat. No.: HY-W009602
CAS No.: 3918-87-4
Synonyms: Phe-ala
Phenylalanylalanine (Phe-ala) is an enkephalinase inhibitor and belongs to the class of dipeptides. Phenylalanylalanine inhibits dipeptidyl carboxypeptidase-mediated enkephalin degradation by cleaving the Gly3-Phe4 bond, and when co-administered with Leu-enkephalin, it produces analgesic effects with a synergistic enhancement, which can be reversed by Naloxone (HY-17417A). Phenylalanylalanine can be used in pain-related research .
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Cat. No.: HY-113278
CAS No.: 3063-05-6
Purity:  99.56%
Leucyl-phenylalanine is a linear dipeptide composed of L-leucine and L-phenylalanine, and also serves as a cyclization substrate. Leucyl-phenylalanine is an incomplete degradation product generated during protein breakdown or catabolism. Leucyl-phenylalanine undergoes heat-induced solid-state cyclization via an autocatalytic mechanism to form its cyclic diketopiperazine analog .
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Cat. No.: HY-101402A
CAS No.: 936749-56-3
Purity:  99.06%
Synonyms: Cyclohistidyl-proline TFA; Histidylproline diketopiperazine TFA
Cyclo(his-pro) TFA (Cyclo(histidyl-proline) TFA) is an orally active cyclic dipeptide structurally related to tyreotropin-releasing hormone . Cyclo(his-pro) TFA could inhibit NF-κB nuclear accumulation. Cyclo(his-pro) TFA can cross the brain-blood-barrier and affect diverse inflammatory and stress responses .
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Cat. No.: HY-107091
CAS No.: 110954-19-3
Purity:  98.87%
Synonyms: DA-DKP
Target:  

Endogenous Metabolite

Research Areas:  

Inflammation/Immunology

Aspartyl-alanyl-diketopiperazine (DA-DKP) is an immunomodulatory molecule generated by cleavage and cyclization from the N-terminus of human albumin and can modulate the inflammatory immune response through a molecular pathway implicated in T- lymphocyte anergy .
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Cat. No.: HY-N8548
CAS No.: 175414-35-4
Fellutanine A, a diketopiperazine alkaloid, is a fungal metabolite from cultures of Penicillium fellutanum .
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Cat. No.: HY-P3472
CAS No.: 57089-60-8
Synonyms: Cyclo(L-Pro-L-Ile)
Research Areas:  

Inflammation/Immunology

Cyclo(IP) (Cyclo-(L-Pro-L-Ile)), a Diketopiperazine can be derived From Bacillus thuringiensis JCK-1233, results in suppression of PWD severity and increased the expression of defense-related genes similarly to Bacillus thuringiensis JCK-1233 treatment .
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Cat. No.: HY-142075
CAS No.: 14474-71-6
Antibacterial agent 134 is the major metabolite in the culture of Hymeniacidon perleve associated bioactive bacterium Pseudomonas sp. NJ6-3-1. Antibacterial agent 134 can be used for bacterial infection .
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Cat. No.: HY-113278S
Leucyl-phenylalanine- 13C6, 15N TFA is the 13C, 15N-labeled Leucyl-phenylalanine (HY-113278). Leucyl-phenylalanine is a linear dipeptide composed of L-leucine and L-phenylalanine, and also serves as a cyclization substrate. Leucyl-phenylalanine is an incomplete degradation product generated during protein breakdown or catabolism. Leucyl-phenylalanine undergoes heat-induced solid-state cyclization via an autocatalytic mechanism to form its cyclic diketopiperazine analog .
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Cat. No.: HY-118100
CAS No.: 21754-25-6
Synonyms: Cyclo(L-Tyr-L-Val)
Target:  

Drug Metabolite

Research Areas:  

Others

Cyclo(Tyr-Val) (Cyclo(L-Tyr-L-Val)) is a diketopiperazine secondary fungal metabolite originally isolated from N. gilva.
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Cat. No.: HY-137361
CAS No.: 108736-10-3
Synonyms: Ramipril diketopiperazine acid
Ramiprilat diketopiperazine (Ramipril diketopiperazine acid; Impurity K) is an impurity of Ramiprilat (HY-A0115). Ramiprilat, an active metabolite of Ramipril (HY-B0279), is a potent and orally active angiotensin converting enzyme (ACE) inhibitor .
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Cat. No.: HY-Z8381
CAS No.: 108731-95-9
Ramipril diketopiperazine is an impurity in the ACE inhibitor Ramipril (HY-B0279) .
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Cat. No.: HY-N12900
CAS No.: 55062-34-5
Synonyms: Tryptophandehydrobutyrine diketopiperazine
TDD (Tryptophandehydrobutyrine diketopiperazine) is a mold metabolite and can be isolated from Streptomyces spectabilis .
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Cat. No.: HY-114547
CAS No.: 103733-49-9
Synonyms: Quinapril diketopiperazine
Target:  

Drug Metabolite

Research Areas:  

Others

PD 109488 is a quinapril diketopiperazine metabolite .
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Cat. No.: HY-114547R
CAS No.: 103733-49-9
Synonyms: Quinapril diketopiperazine (Standard)
Research Areas:  

Others

PD 109488 (Standard) is the analytical standard of PD 109488. This product is intended for research and analytical applications. PD 109488 is a quinapril diketopiperazine metabolite .
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Cat. No.: HY-N10222
CAS No.: 871982-52-4
Roquefortine E is a diketopiperazine from an Australian isolate of Gymnoascus reessii .
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Cat. No.: HY-N8513
CAS No.: 215121-47-4
Brevicompanine B, a diketopiperazine alkaloid, is an antiplasmodial agent. Brevicompanine B is active against the malaria parasite Plasmodium falciparum 3D7 IC50 of 35 mg/mL .
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Cat. No.: HY-90009R
CAS No.: 171596-36-4
Synonyms: Demethyl Tadalafil (Standard)
Nortadalafil (Standard) is the analytical standard of Nortadalafil. This product is intended for research and analytical applications. Nortadalafil , a new tadalafil (HY-90009A) analogue detected in health foods, is a PDE5 inhibitor. Nortadalafil is used in the research of erectile dysfunction (ED). Nortadalafil can be formed by closing the diketopiperazine ring in high yield. Nortadalafil is promising for research of pulmonary arterial hypertension [4] .
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