3 Results for "

lyso-PAF/acetyl-CoA acetyltransferase

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "lyso-PAF/acetyl-CoA acetyltransferase" in MCE Product Catalog:

Cat. No.: HY-112825
CAS No.: 704878-75-1
Purity:  98.52%
Research Areas:  

Inflammation/Immunology Cancer

TSI-01 is a selective LPCAT2 inhibitor, with IC50 values of 0.47 μM and 3.02 μM against LPCAT2 and LPCAT1, respectively. TSI-01 competitively inhibits acetyl-CoA (acetyl-CoA) targeting the lysophosphatidic acid acetyltransferase activity of LPCAT2, and suppresses PAF biosynthesis in calcium ionophore-stimulated mouse peritoneal macrophages. TSI-01 inhibits the proliferation of endometrial cancer cells and promotes endometrial cancer cell apoptosis (apoptosis). TSI-01 can be used for the research of endometrial cancer and PAF-related inflammatory diseases .
loading...
    loading...
Cat. No.: HY-P811936
Synonyms: AGPAT11, AYTL1, LPCAT2, lysophosphatidylcholine acyltransferase 2, LPC acyltransferase 2, LPCAT-2, lysoPC acyltransferase 2, 1-acylglycerol-3-phosphate O-acyltransferase 11, 1-acylglycerophosphocholine O-acyltransferase, 1-alkenylglycerophosphocholine O-acyltransferase, 1-alkylglycerophosphocholine O-acetyltransferase, acetyl-CoA:lyso-platelet-activating factor acetyltransferase, Acyltransferase-like 1, lysophosphatidic acid acyltransferase alpha, 1-AGP acyltransferase 11, 1-AGPAT 11, acetyl-CoA:lyso-PAF acetyltransferase, lyso-PAF acetyltransferase, lysoPAFAT, LPAAT-alpha

Host:  

Mouse

Application:  

WB, FC, ICC/IF

Reactivity:  

Human

loading...
    loading...
Cat. No.: HY-P811936A
Synonyms: AGPAT11, AYTL1, LPCAT2, lysophosphatidylcholine acyltransferase 2, LPC acyltransferase 2, LPCAT-2, lysoPC acyltransferase 2, 1-acylglycerol-3-phosphate O-acyltransferase 11, 1-acylglycerophosphocholine O-acyltransferase, 1-alkenylglycerophosphocholine O-acyltransferase, 1-alkylglycerophosphocholine O-acetyltransferase, acetyl-CoA:lyso-platelet-activating factor acetyltransferase, Acyltransferase-like 1, lysophosphatidic acid acyltransferase alpha, 1-AGP acyltransferase 11, 1-AGPAT 11, acetyl-CoA:lyso-PAF acetyltransferase, lyso-PAF acetyltransferase, lysoPAFAT, LPAAT-alpha

Host:  

Mouse

Application:  

WB, FC, ICC/IF

Reactivity:  

Human

loading...
    loading...