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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
20 Results for "
tricyclic compound
" in MedChemExpress (MCE) Product Catalog:
Products (20)
20 Results for "tricyclic compound" in MCE Product Catalog:
Cat. No.: HY-136645
CAS No.: 1965316-82-8
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EP4 receptor antagonist 2 (Compound 8) is a tricyclic spiro-based EP4 receptor antagonist with microsomal stability .
Cat. No.: HY-44745
CAS No.: 127318-97-2
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Camptothecin impurity 1 (Compound 1) is an impurity of Camptothecin (HY-16560), which serves as a starting compound for the synthesis of tricyclic intermediates of Camptothecin .
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Dibenzosuberone is a tricyclic compound, commonly referred to as a tricyclic antidepressant (TCA), and is widely used in research on migraine, tension-type headache, anxiety disorder and schizophrenia. Dibenzosuberone also serves as a key intermediate for the synthesis of various active pharmaceutical ingredients (APIs) (e.g., amitriptyline (HY-B0527), nortriptyline (HY-118620), nortriptyline or cyproheptadine (HY-B1622)) .
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BRD0209 is a potent, selective and dual inhibitor of GSK3α/β inhibitor (GSK3α IC50 = 19 nM; GSK3β IC50 = 5 nM). BRD0209 is also a reversible ATP-competitive inhibitor with fast-off kinetics (Ki = 4.2 nM, respectively). BRD0209 is a tricyclic pyrazolotetrahydroquinolinone compound. BRD0209 has the potential for the research of mood disorder diseases .
Cat. No.: HY-19773
CAS No.: 1075237-97-6
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β-Lactamase-IN-1 is an inhibitor of β-Lactamase extracted from patent WO2016027249A1, page 77. β-Lactamase-IN-1 can be used to prepare of tricyclic nitrogen containing compound. β-Lactamase-IN-1 can be used for the research of neisseria gonorrhea infection .
Cat. No.: HY-151500C
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JBSNF-00002 is an orally active small molecule inhibitor of the tricyclic nicotinamide N-methyltransferase (NNMT) with IC50 values for human, mouse and monkey sources of NNMT of 33, 210 and 190 nM respectively. JBSNF-00002 can reduce endogenous MNA levels in U2OS osteosarcoma cells, with its EC50 being 2.5 μM. JBSNF-00002 exhibits significant anti-obesity and anti-diabetic activities in the diet-induced obesity (DIO) model. JBSNF-00002 can be used for the study of metabolic diseases such as obesity, type 2 diabetes and non-alcoholic fatty liver disease .
Cat. No.: HY-161878
CAS No.: 2857051-98-8
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USP1-IN-10 (compound 2) is a potent tricyclic USP1 inhibitor with an IC50 of 7.6 nM. USP1-IN-10 inhibits MDA-MB-436 viability (IC50=21.58 nM). USP1-IN-10 has the potential for cancers research .
Cat. No.: HY-179275
CAS No.: 3099165-43-9
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TLR7 agonist 33 (Compound 141) is a potent TLR7 activator with an EC50 of 1 nM. TLR7 agonist 33 can be used for cancer research .
Cat. No.: HY-106079
CAS No.: 80410-36-2
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Fezolamine is an orally active non-tricyclic compound , and shows antidepressant activity .
Cat. No.: HY-N13178
CAS No.: 157744-28-0
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Cat. No.: HY-N11977
CAS No.: 208834-81-5
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Cat. No.: HY-44745S
CAS No.: 1346605-23-9
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Camptothecin impurity 1-d5 is the d5-labeled Camptothecin impurity 1 (HY-44745). Camptothecin impurity 1 (Compound 1) is an impurity of Camptothecin (HY-16560), which serves as a starting compound for the synthesis of tricyclic intermediates of Camptothecin .
Cat. No.: HY-107031
CAS No.: 21730-16-5
Synonyms: 19560 RP
Metapramine (19560 RP) is an antidepressant agent, belonging to the class of tricyclic compounds . Metapramine inhibits norepinephrine reuptake, without affecting the reuptake of serotonin or dopamine . Metapramine is a low-affinity antagonist of the N-methyl-D-aspartic acid (NMDA) receptor complex channel .
Cat. No.: HY-114604
CAS No.: 102962-95-8
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Cat. No.: HY-175194
CAS No.: 2755671-89-5
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5-HT2C agonist-6 (Compound 13), a tricyclic psychedelic psychoplastogen, is a 5-HT2C agonist with an EC50 of 13.8 nM. 5-HT2C agonist-6 can be used for neurological diseases research .
Cat. No.: HY-167672
CAS No.: 10321-12-7
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Propizepine is a tricyclic antidepressant compound .
Cat. No.: HY-184039
CAS No.: 88124-26-9
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Adosupine is a tricyclic compound that affects detrusor hyperreflexia via central nervous system sites. Adosupine can be used in studies related to detrusor hyperreflexia and urinary incontinence .
Cat. No.: HY-44745R
CAS No.: 127318-97-2
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Camptothecin impurity 1 (Standard) is the analytical standard of Camptothecin impurity 1 (HY-44745). This product is intended for research and analytical applications. Camptothecin impurity 1 (Compound 1) is an impurity of Camptothecin (HY-16560), which serves as a starting compound for the synthesis of tricyclic intermediates of Camptothecin .
Cat. No.: HY-W609889
CAS No.: 1239879-65-2
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5-HT2A receptor agonist-14 (Compound I-23) is a tricyclic 5-HT2A receptor agonist with a pEC50 value ≥ 6. 5-HT2A receptor agonist-14 can be used in research related to depression, anxiety, substance abuse and headache .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
