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  2. Estrogen Receptor/ERR
  3. ERRγ Inverse Agonist 1

ERRγ Inverse Agonist 1 

Cat. No.: HY-114411
Handling Instructions

ERRγ Inverse Agonist 1 (Compound 12) is a potent, selective and orally bioavailable Estrogen-related Receptor grammar (ERRγ) inverse agonist, with an IC50 of 40 nM.

For research use only. We do not sell to patients.

ERRγ Inverse Agonist 1 Chemical Structure

ERRγ Inverse Agonist 1 Chemical Structure

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Description

ERRγ Inverse Agonist 1 (Compound 12) is a potent, selective and orally bioavailable Estrogen-related Receptor grammar (ERRγ) inverse agonist, with an IC50 of 40 nM[1].

IC50 & Target[1]

ERRγ

0.040 μM (IC50)

ERRβ

1.330 μM (IC50)

ERα

1.240 μM (IC50)

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
Molecular Weight

529.54

Formula

C₃₀H₃₈Cl₂N₂O₂

SMILES

OC1=CC=CC(/C(C2=CC=C(N3CCN(C(C)C)CC3)C=C2)=C(C4=CC=CC=C4)\CCCO)=C1.[H]Cl.[H]Cl

Shipping

Room temperature in continental US; may vary elsewhere

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  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Product Name:
ERRγ Inverse Agonist 1
Cat. No.:
HY-114411
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ERRγ Inverse Agonist 1

Cat. No.: HY-114411