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  2. Estrogen Receptor/ERR
  3. ERRγ Inverse Agonist 1

ERRγ Inverse Agonist 1 

Cat. No.: HY-114411
Handling Instructions

ERRγ Inverse Agonist 1 (Compound 12) is a potent, selective and orally bioavailable Estrogen-related Receptor grammar (ERRγ) inverse agonist, with an IC50 of 40 nM.

For research use only. We do not sell to patients.

ERRγ Inverse Agonist 1 Chemical Structure

ERRγ Inverse Agonist 1 Chemical Structure

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Description

ERRγ Inverse Agonist 1 (Compound 12) is a potent, selective and orally bioavailable Estrogen-related Receptor grammar (ERRγ) inverse agonist, with an IC50 of 40 nM[1].

IC50 & Target[1]

ERRγ

0.040 μM (IC50)

ERRβ

1.330 μM (IC50)

ERα

1.240 μM (IC50)

Molecular Weight

529.54

Formula

C₃₀H₃₈Cl₂N₂O₂

SMILES

OC1=CC=CC(/C(C2=CC=C(N3CCN(C(C)C)CC3)C=C2)=C(C4=CC=CC=C4)\CCCO)=C1.[H]Cl.[H]Cl

Shipping

Room temperature in continental US; may vary elsewhere

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
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Product Name:
ERRγ Inverse Agonist 1
Cat. No.:
HY-114411
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