GHSR Antagonist
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JMV 2959
0 ImagesJMV 2959 is a growth hormone secretagogue receptor type 1a (GHS-R1a) antagonist with an IC50 of 32 nM.
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JMV 2959 hydrochloride
0 ImagesCat. No.: HY-U00433ACAS No.: 2448414-54-6JMV 2959 hydrochloride is a growth hormone secretagogue receptor type 1a (GHS-R1a) antagonist with an IC50 of 32±3 nM in LLC-PK1 cells.
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Acetyl-(D-Arg2)-GRF (1-29) amide (human)
0 ImagesAcetyl-(D-Arg2)-GRF (1-29) amide (human) is an antagonist of growth hormone releasing factor (GRF). Acetyl-(D-Arg2)-GRF (1-29) amide (human) inhibits the release of growth hormone (GH) and can be used for endocrine research.
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GSK1614343
0 ImagesCat. No.: HY-113906CAS No.: 1092076-04-4GSK1614343 is the potent antagonist of growth hormone secretagogues type 1a (GHS1a) receptors. GSK1614343 inhibits the calcium response induced by ghrelin with a pIC50 value of 7.90. GSK1614343 represents a useful tool to investigate the physiological relevance of the ghrelin system in rat models.
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AZ-GHS-22
0 ImagesCat. No.: HY-137061CAS No.: 1143020-91-0AZ-GHS-22 is a potent, non-CNS penetrant GHS-R1a inverse agonist (IC50=0.77 nM).
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K-(D-1-Nal)-FwLL-NH2
0 ImagesCat. No.: HY-P1432CAS No.: 1394288-22-2K-(D-1-Nal)-FwLL-NH2 is a high affinity, potent and inverse ghrelin receptor agonist (EC50=3.4 nM, Ki=4.9 nM). K-(D-1-Nal)-FwLL-NH2 can be used for the research of obesity.
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Tezusomant
0 ImagesCat. No.: HY-P10964CAS No.: 2802416-72-2Tezusomant is a growth hormone receptor antagonist. Tezusomant is promising for research on diseases caused by excessive growth hormone secretion, such as acromegaly.
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KwFwLL-NH2
0 ImagesCat. No.: HY-P10673CAS No.: 942266-38-8KwFwLL-NH2, a hexapeptide, is a ghrelin receptor ligand. KwFwLL-NH2 can act as a specific inverse agonist at the ghrelin receptor but with moderate potency (EC50=45.6 nM).
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