1092076-04-4
Chemical Structure
GSK1614343
- CAS No.: 1092076-04-4
- Formula:C22H23F6N5O
- Molecular Weight:487.44
IUPAC Name: (R)-N'-(3,5-bis(trifluoromethyl)phenyl)-2-((R)-hexahydropyrrolo[1,2-a]pyrazin-2(1H)-yl)-2-(pyridin-3-yl)acetohydrazide
InChIKey: QNOSCJDGJKVFJR-RTBURBONSA-N
SMILES: O=C([C@@H](C1=CC=CN=C1)N2C[C@@]3([H])CCCN3CC2)NNC4=CC(C(F)(F)F)=CC(C(F)(F)F)=C4
Biological Activity: GSK1614343 is the potent antagonist of growth hormone secretagogues type 1a (GHS1a) receptors. GSK1614343 inhibits the calcium response induced by ghrelin with a pIC50 value of 7.90. GSK1614343 represents a useful tool to investigate the physiological relevance of the ghrelin system in rat models[1].
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GSK1614343 | GSK1614343 is the potent antagonist of growth hormone secretagogues type 1a (GHS1a) receptors. GSK1614343 inhibits the calcium response induced by ghrelin with a pIC50 value of 7.90. GSK1614343 represents a useful tool to investigate the physiological relevance of the ghrelin system in rat models. | |||||||||||||||||||||
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