Neurotensin Receptor Activator
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[Lys8, Lys9]-Neurotensin (8-13)
![[Lys8, Lys9]-Neurotensin (8-13)](https://file.medchemexpress.com/product_pic/hy-p2544.gif "Click to View [Lys8, Lys9]-Neurotensin (8-13) Product Detail")
0 ImagesSynonyms: JMV438[Lys8, Lys9]-Neurotensin (8-13) (JMV438), a Neurotensin analog, exerts its analgesic effects through activation of the G protein-coupled receptors NTS1 and NTS2, with Ki values of 0.33 nM and 0.95 nM for hNTS1 and hNTS2 receptors, respectively.
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MD01-67
0 ImagesCat. No.: HY-P10767CAS No.: 2468971-42-6MD01-67 is a selective macrocyclic compound targeting the neurotensin receptor type 2 (NTS2), with Ki of 2.9 nM. MD01-67 exhibits analgesic and tactile hypersensitivity reducing activity in rats acute/persistent/chronic inflammatory pain models.
