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Cat. No.: HY-162125

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AT2 receptor ligand-1

AT2 receptor ligand-1(compound 14) is a potent angiotensin AT2 receptor ligand with the K_i 4.9 nM. AT2 receptor ligand-1 shows high stability in microsomes of the sulfonamide ligands.

For research use only. We do not sell to patients.

CAS No.: 3027141-86-9

Formula: C₂₇H₃₁N₅O₃S₂

Molecular Weight:537.70

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (273 KB)

AT2 receptor ligand-1 Chemical Structure

CAS No.: 3027141-86-9

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Data Sheet (273 KB)

Handling Instructions (2659 KB)

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Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

All Angiotensin Receptor Isoforms
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AT1 Receptor

AT2 Receptor

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Bioz

Biological Activity

Description

AT2 receptor ligand-1(compound 14) is a potent angiotensin AT2 receptor ligand with the K_i 4.9 nM. AT2 receptor ligand-1 shows high stability in microsomes of the sulfonamide ligands^[1].

All Angiotensin Receptor Isoforms :

AT1 Receptor

AT2 Receptor

Chemical Information

CAS No. 3027141-86-9

Molecular Weight 537.70

Formula C₂₇H₃₁N₅O₃S₂

SMILES

O=S(C1=C(C2=CC=CC(C(CN3C=CN=C3C(C)(C)C)=O)=C2)C=C(CC(C)C)S1)(NC4=NC=CC=N4)=O

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (273 KB)

COA (2659 KB)

Elemental Analysis Report (2659 KB)

HNMR (2659 KB)

CNMR (2659 KB)

RP-HPLC (2659 KB)

NP-HPLC (2659 KB)

MS (2659 KB)

LCMS (2659 KB)

IR (2659 KB)

GC (2659 KB)

OR (2659 KB)

SDS-PAGE (2659 KB)

SEC-HPLC (2659 KB)

Other Report (2659 KB)

Handling Instructions (2659 KB)

References

[1]. Wannberg J, et al. N-(Heteroaryl)thiophene sulfonamides as angiotensin AT2 receptor ligands. Eur J Med Chem. 2024;265:116122. [Content Brief]

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How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

AT2 receptor ligand-1 Related Classifications

HY-162125 Related Classifications

GPCR/G Protein

Angiotensin Receptor

Disease Areas

Blood or Cardio-cerebrovascular Disease

Cardiovascular Disease

Powered by Bioz See more details on Bioz

Keywords

AT2 receptor ligand-1
3027141-86-9
Angiotensin Receptor
Angiotensin II type 2 receptor
AT2R ligands
N-heteroaryl sulfonamides
Carboxylic acid bioisosteres
Inhibitor
inhibitor
inhibit

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ナミキ商事株式会社コスモ・バイオ株式会社重松貿易株式会社

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