100111-08-8
100111-08-8
Chemical Structure
H256
- CAS No.: 100111-08-8
- Formula:C43H62N10O12
- Molecular Weight:911.01
IUPAC Name: (2-(4-carboxy-2-(3-hydroxy-2-(pyrrolidine-2-carboxamido)butanamido)butanamido)-3-phenylpropyl)phenylalanylarginylglutamic acid
InChIKey: WNWJVPXOYQRRNI-MVPDBZEZSA-N
SMILES: O=C(O)CC[C@@H](C(O)=O)NC([C@H](CCCNC(N)=N)NC([C@H](CC1=CC=CC=C1)NC[C@@H](NC([C@H](CCC(O)=O)NC([C@H]([C@H](O)C)NC([C@H]2NCCC2)=O)=O)=O)CC3=CC=CC=C3)=O)=O
Biological Activity: H256 is an inhibitor of Endothiapepsin and Pepsin, with a Ki value of 60 nM against Endothiapepsin[1][2].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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H256 | H256 is an inhibitor of Endothiapepsin and Pepsin, with a Ki value of 60 nM against Endothiapepsin. | |||||||||||||||||||||
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References
- [1]. Cooper J, et al. The structure of a synthetic pepsin inhibitor complexed with endothiapepsin. Eur J Biochem. 1987 Nov 16;169(1):215-21.
- [2]. Guruprasad K, et al. Comparative modelling of barley-grain aspartic proteinase: a structural rationale for observed hydrolytic specificity. FEBS Lett. 1994 Sep 26;352(2):131-6.
