1049691-47-5
1049691-47-5
Chemical Structure
NR2F2-IN-1
- CAS No.: 1049691-47-5
- Formula:C17H20ClN3O2S
- Molecular Weight:365.88
InChIKey: PYRMFONFWQTEGD-UHFFFAOYSA-N
SMILES: COC(C(OC)=C1)=CC=C1CCNC2=C3C=C(C)SC3=NC=N2.Cl
Biological Activity: NR2F2-IN-1 (COUP-TFII inhibitor) is a small-molecule inhibitor targeting the orphan nuclear receptor COUP-TFII (NR2F2). NR2F2-IN-1 directly binds to the ligand-binding domain of COUP-TFII (NR2F2) and disrupts its interaction with transcriptional regulators including FOXA1. NR2F2-IN-1 induces anti-tumor activity in prostate cancer and can be used for prostate cancer research[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
|
|
NR2F2-IN-1 | NR2F2-IN-1 (COUP-TFII inhibitor) is a small-molecule inhibitor targeting the orphan nuclear receptor COUP-TFII (NR2F2). NR2F2-IN-1 directly binds to the ligand-binding domain of COUP-TFII (NR2F2) and disrupts its interaction with transcriptional regulators including FOXA1. NR2F2-IN-1 induces anti-tumor activity in prostate cancer and can be used for prostate cancer research. | |||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
References
Keywords
