120770-34-5
Chemical Structure
Draflazine
Synonym(s): R-75231; R88021
- CAS No.: 120770-34-5
- Formula:C30H33Cl2F2N5O2
- Molecular Weight:604.52
IUPAC Name: 1-(2-((4-amino-2,6-dichlorophenyl)amino)-2-oxoethyl)-4-(5,5-bis(4-fluorophenyl)pentyl)piperazine-2-carboxamide
InChIKey: IWMYIWLIESDFRZ-UHFFFAOYSA-N
SMILES: O=C(NC1=C(Cl)C=C(N)C=C1Cl)CN2C(C(N)=O)CN(CCCCC(C3=CC=C(F)C=C3)C4=CC=C(F)C=C4)CC2
Biological Activity: Draflazine (R-75231) is a ENT1 inhibitor. Draflazine (R-75231) completely reverses the hypersensitivity in the complete Freund’s adjuvant (CFA) model of mechanical hyperalgesia and the carrageenan inflammation model of thermal and mechanical hyperalgesia[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Draflazine | 99.06% | Draflazine (R-75231) is a ENT1 inhibitor. Draflazine (R-75231) completely reverses the hypersensitivity in the complete Freund’s adjuvant (CFA) model of mechanical hyperalgesia and the carrageenan inflammation model of thermal and mechanical hyperalgesia. | ||||||||||||||||||||
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Similarity Score 1.00
HY-106841A(S)-Draflazine -
Similarity Score 0.80
HY-U00049Mioflazine -
Similarity Score 0.80
HY-U00049BMioflazine dihydrochloride -
Similarity Score 0.80
HY-U00049AMioflazine (di(hydrochloride) hydrate) -
Similarity Score 0.70
HY-115366Soluflazine -
Similarity Score 0.63
HY-112075Lidoflazine -
Similarity Score 0.56
HY-W2491081-(4,4-Bis(4-fluorophenyl)butyl)-4-(4-chloro-3-(trifluoromethyl)phenyl)piperidin-4-ol acetate -
Similarity Score 0.55
HY-121301Amperozide -
Similarity Score 0.55
HY-B1077Penfluridol -
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