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Draflazine (Synonyms: R-75231)

Cat. No.: HY-106841
Handling Instructions

Draflazine (R-75231) is a ENT1 inhibitor. Draflazine (R-75231) completely reverses the hypersensitivity in the complete Freund’s adjuvant (CFA) model of mechanical hyperalgesia and the carrageenan inflammation model of thermal and mechanical hyperalgesia.

For research use only. We do not sell to patients.

Draflazine Chemical Structure

Draflazine Chemical Structure

CAS No. : 120770-34-5

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Description

Draflazine (R-75231) is a ENT1 inhibitor. Draflazine (R-75231) completely reverses the hypersensitivity in the complete Freund’s adjuvant (CFA) model of mechanical hyperalgesia and the carrageenan inflammation model of thermal and mechanical hyperalgesia[1].

IC50 & Target

ENT1[1]

Molecular Weight

604.52

Formula

C₃₀H₃₃Cl₂F₂N₅O₂

CAS No.

120770-34-5

SMILES

O=C(NC1=C(Cl)C=C(N)C=C1Cl)CN2C(C(N)=O)CN(CCCCC(C3=CC=C(F)C=C3)C4=CC=C(F)C=C4)CC2

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Room temperature in continental US; may vary elsewhere

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Draflazine
Cat. No.:
HY-106841
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