1418308-27-6
1418308-27-6
Chemical Structure
EI1
Synonym(s): KB-145943
- CAS No.: 1418308-27-6
- Formula:C23H26N4O2
- Molecular Weight:390.48
IUPAC Name: 6-cyano-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-1-(pentan-3-yl)-1H-indole-4-carboxamide
InChIKey: PFHDWRIVDDIFRP-UHFFFAOYSA-N
SMILES: CCC(CC)N(C=C1)C2=C1C(C(NCC3=C(C)C=C(C)NC3=O)=O)=CC(C#N)=C2
Biological Activity: EI1 (KB-145943) is a potent and selective EZH2 inhibitor with IC50 of 15 nM and 13 nM for EZH2 (WT) and EZH2 (Y641F), respectively.
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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EI1 | 98.84% | EI1 (KB-145943) is a potent and selective EZH2 inhibitor with IC50 of 15 nM and 13 nM for EZH2 (WT) and EZH2 (Y641F), respectively. | ||||||||||||||||||||
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Keywords
