144625-51-4
144625-51-4
Chemical Structure
GR 113808
- CAS No.: 144625-51-4
- Formula:C19H27N3O4S
- Molecular Weight:393.50
IUPAC Name: (1-(2-(methylsulfonamido)ethyl)piperidin-4-yl)methyl 1-methyl-1H-indole-3-carboxylate
InChIKey: MOZPSIXKYJUTKI-UHFFFAOYSA-N
SMILES: O=C(C1=CN(C)C2=C1C=CC=C2)OCC3CCN(CCNS(=O)(C)=O)CC3
Biological Activity: GR 113808 is a potent and highly selective 5-HT4 receptor antagonist (pKb= 8.8). GR 113808 shows 300-fold selectivity over 5-HT1A, 5-HT1B, 5-HT2A, 5-HT2C and 5-HT3 receptors[1].
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GR 113808 | 99.68% | GR 113808 is a potent and highly selective 5-HT4 receptor antagonist (pKb= 8.8). GR 113808 shows 300-fold selectivity over 5-HT1A, 5-HT1B, 5-HT2A, 5-HT2C and 5-HT3 receptors. | ||||||||||||||||||||
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GR 113808 (Standard) | ≥98% | GR 113808 (Standard) is the analytical standard of GR 113808. This product is intended for research and analytical applications. GR 113808 is a potent and highly selective 5-HT4 receptor antagonist (pKb= 8.8). GR 113808 shows 300-fold selectivity over 5-HT1A, 5-HT1B, 5-HT2A, 5-HT2C and 5-HT3 receptors. | ||||||||||||||||||||
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References
Keywords
