148565-09-7
148565-09-7
Chemical Structure
KB R6933
Synonym(s): KB 6806 maleate
- CAS No.: 148565-09-7
- Formula:C23H30ClN5O8
- Molecular Weight:539.97
InChIKey: ZEYGAOFLBIEQJQ-SPIKMXEPSA-N
SMILES: OC(/C=C\C(O)=O)=O.CC(N1C(N2CCN(CC2)C)=NC3=CC(Cl)=C(N)C=C31)C.OC(/C=C\C(O)=O)=O
Biological Activity: KB R6933 (KB 6806 maleate) is a potent, selective and orally active 5-HT3 receptor antagonist. KB R6933 can inhibit the diarrhea induced by 5-HT (HY-B1473A), but not that by Castor Oil (HY-107799) or prostaglandin E2 (PGE2) (HY-101952). KB R6933 can inhibit 5-HT-induced bradycardia[1][2].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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KB R6933 | KB R6933 (KB 6806 maleate) is a potent, selective and orally active 5-HT3 receptor antagonist. KB R6933 can inhibit the diarrhea induced by 5-HT (HY-B1473A), but not that by Castor Oil (HY-107799) or prostaglandin E2 (PGE2) (HY-101952). KB R6933 can inhibit 5-HT-induced bradycardia. | |||||||||||||||||||||
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References
Keywords
