1637770-13-8
1637770-13-8
Chemical Structure
GS-626510
- CAS 番号: 1637770-13-8
- Formula:C25H22N4O
- Molecular Weight:394.47
IUPAC Name: 4-(2-cyclopropyl-7-(6-methylquinolin-5-yl)-1H-benzo[d]imidazol-5-yl)-3,5-dimethylisoxazole
InChIKey: KHQQNXFBTALTQF-UHFFFAOYSA-N
SMILES: CC1=C(C2=CC(C3=C4C=CC=NC4=CC=C3C)=C5NC(C6CC6)=NC5=C2)C(C)=NO1
Biological Activity: GS-626510 is a potent, and orally active BET family bromodomains inhibitor, with Kd values of 0.59-3.2 nM for BRD2/3/4, with IC50 values of 83 nM and 78 nM foe BD1 and BD2, respectively[1].
| 製品番号 | 製品名 | 純度 | 製品説明 | Pricing | |||||||||||||||||||
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GS-626510 | 99.46% | GS-626510 is a potent, and orally active BET family bromodomains inhibitor, with Kd values of 0.59-3.2 nM for BRD2/3/4, with IC50 values of 83 nM and 78 nM foe BD1 and BD2, respectively. | ||||||||||||||||||||
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References
Keywords
