2445335-77-1
2445335-77-1
Chemical Structure
Bromodomain IN-2
- CAS No.: 2445335-77-1
- Formula:C16H17ClN2O
- Molecular Weight:288.77
IUPAC Name: 1-(5-amino-2-chlorophenyl)-3-methyl-5,6,7,8-tetrahydrocyclohepta[c]pyrrol-4(2H)-one
InChIKey: DGJREYHVQYZTEV-UHFFFAOYSA-N
SMILES: O=C1C2=C(C)NC(C3=C(Cl)C=CC(N)=C3)=C2CCCC1
Biological Activity: BD-IN-1 is a pan bromodomain (BD) inhibitor with KD values of 250, 420, 130, 430, 67, 240, 970 nM for BRD4(1), CBP, BRPF1B, BRD7, BRD9, BRDT(1), CECR2 respectively. BD-IN-1 shows antiproliferative activity[1].
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Bromodomain IN-2 | BD-IN-1 is a pan bromodomain (BD) inhibitor with KD values of 250, 420, 130, 430, 67, 240, 970 nM for BRD4(1), CBP, BRPF1B, BRD7, BRD9, BRDT(1), CECR2 respectively. BD-IN-1 shows antiproliferative activity. | |||||||||||||||||||||
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References
Keywords
