3057089-47-8
3057089-47-8
Chemical Structure
IV-255
- CAS No.: 3057089-47-8
- Formula:C19H19F2N3O2
- Molecular Weight:359.37
InChIKey: LUTFUXGPBODRIB-HUUCEWRRSA-N
SMILES: COC1=CC=C(N2[C@H]3CN([C@@H](C2)C3)C(NC4=CC(F)=C(C=C4)F)=O)C=C1
Biological Activity: IV-255 is a selective small molecule inhibitor of the BRG1 bromodomain. IV-255 increases the extent of DNA damage induced by Temozolomide (HY-17364) and Bleomycin (HY-108345). IV-255 inhibits the invasiveness of GBM cells. IV-255 enhances Temozolomide-induced cell death and the apoptosis-inducing activity of Temozolomide[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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IV-255 | 99.28% | IV-255 is a selective small molecule inhibitor of the BRG1 bromodomain. IV-255 increases the extent of DNA damage induced by Temozolomide (HY-17364) and Bleomycin (HY-108345). IV-255 inhibits the invasiveness of GBM cells. IV-255 enhances Temozolomide-induced cell death and the apoptosis-inducing activity of Temozolomide. | ||||||||||||||||||||
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