CK1δ-IN-9
CK1δ-IN-9 (Compound 8) is the inhibitor for casein kinase 1 that inhibits CK1δ with IC50 of 1.4 nM. CK1δ-IN-9 inhibits p38α and p38β with IC50 of 0.25 μM and 0.78 μM. CK1δ-IN-9 exhibits pharmacokinetic characteristics with a good oral bioavailability (70%) and a moderate clearance.
For research use only. We do not sell to patients.
- CAS No.: 3057263-82-5
- Formula: C16H12FN5
- Molecular Weight:293.30
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
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CK1δ 1.4 nM (IC50) |
p38α 0.25 μM (IC50) |
p38β 0.78 μM (IC50) |
Chemical Information
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CAS No. 3057263-82-5
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Molecular Weight 293.30
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Formula C16H12FN5
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SMILES
FC1=CC=C(C2=NN(C)C=C2C3=C4C=NNC4=NC=C3)C=C1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
CK1δ-IN-9 Related Classifications
HY-171292 Related Classifications
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