2. GPCR/G Protein Neuronal Signaling
  3. Dopamine Receptor
  4. Dopamine D2 receptor agonist-3

Dopamine D2 receptor agonist-3 (compound 3) is a selective D2 receptor partial agonist and Dopamine D3 receptor antagonist (with pEC50 of 8.3 and <5.5 respectively).

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Dopamine D2 receptor agonist-3 Chemical Structure

Dopamine D2 receptor agonist-3 Chemical Structure

CAS No. : 1257326-24-1

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Based on 1 publication(s) in Google Scholar

Dopamine D2 receptor agonist-3 Related Antibodies

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Description

Dopamine D2 receptor agonist-3 (compound 3) is a selective D2 receptor partial agonist and Dopamine D3 receptor antagonist (with pEC50 of 8.3 and <5.5 respectively)[1].

IC50 & Target[1]

D2 Receptor

5 nM (EC50)

D3 Receptor

>3.2 μM (EC50)

In Vivo

Dopamine D2 receptor agonist-3 (3 mg/kg, s.c.) shows high brain penetration (brain to blood ratio of 5.5) and Tmax of 0.5 h[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Molecular Weight

295.81

Formula

C15H22ClN3O
CAS No.
Appearance

Solid

SMILES

O=C1N(CC2NCCCC2)CCN1C3=CC=CC=C3.[H]Cl
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

4°C, protect from light

*In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)

Purity & Documentation
References
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Dopamine D2 receptor agonist-3 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Dopamine D2 receptor agonist-31257326-24-1Dopamine ReceptorDopaminepartial agonistInhibitorinhibitorinhibit

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