Dyrk1A-IN-11
Dyrk1A-IN-11 (compound 166) is a potent dual-specificity tyrosine phosphorylation- regulated 1A (DYRK1A) inhibitor with an EC50 value of 0.0021 µM. Dyrk1A-IN-11 inhibits the Phospho-Tau (Thr212) with an EC50 value of 0.0361 µM.
For research use only. We do not sell to patients.
- CAS No.: 3058626-26-6
- Formula: C23H23F5N8O
- Molecular Weight:522.47
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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DYRK1A 0.0021 μM (EC50) |
Chemical Information
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CAS No. 3058626-26-6
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Molecular Weight 522.47
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Formula C23H23F5N8O
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SMILES
CC1=NC2=C(N1CC(F)F)N=C(C3=C4N(N=C(N[C@@H]5CCN(C6COC6)CC5(F)F)N=C4)C=C3F)C=C2
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)