DYRK Inhibitors

DYRK1

DYRK2

DYRK3

DYRK4

HIPK

PRP4

DYRK Inhibitors & Degraders

Product Name	DYRK1	DYRK2	DYRK3	DYRK4	HIPK	PRP4	Purity
Harmine	DYRK1A						99.97%
AZ191	DYRK1B						99.98%
GNF2133	DYRK1A, IC₅₀: 0.0062 μM						99.67%
DYRK2-IN-2	DYRK1A, IC₅₀: 1842 nM DYRK1B, IC₅₀: 1335 nM	DYRK2, IC₅₀: 40.3 nM	DYRK3, IC₅₀: 112 nM	DYRK4, IC₅₀: 1931 nM
AO-365/43472821	DYRK1A, IC₅₀: 0.29 μM
Harmine hydrochloride	DYRK1A						99.98%
GNF4877	DYRK1A, IC₅₀: 6 nM						99.82%
GSK-626616	DYRK1	DYRK2	DYRK3				99.88%
INDY	DYRK1A DYRK1B						99.32%
T025	DYRK1A, Kd: 0.074 nM DYRK1B, Kd: 1.5 nM	DYRK2, Kd: 32 nM					99.64%
ML167	DYRK1A, IC₅₀: ＞10000 nM DYRK1B, IC₅₀: 4420 nM						98.62%
Protein kinase inhibitor 1 hydrochloride	DYRK1	DYRK2					98.0%
Leucettine L41	DYRK1A, IC₅₀: 10-60 nM DYRK1B, IC₅₀: 44 nM	DYRK2, IC₅₀: 73 nM	DYRK3, IC₅₀: 320 nM	DYRK4, IC₅₀: 520 nM			98.98%
DYRK1-IN-1	DYRK1A, IC₅₀: 220 nM DYRK1A, Kd: 3 nM DYRK1B, Kd: 56 nM						99.71%
RO5454948	DYRK1A, IC₅₀: 22 nM DYRK1B, IC₅₀: 68 nM						99.53%
Dyrk1A-IN-5	DYRK1A, IC₅₀: 6 nM DYRK1B, IC₅₀: 600 nM	DYRK2, IC₅₀: > 10000 nM					98.06%
AZ-Dyrk1B-33	DYRK1B						99.78%
YK-2-69		DYRK2, IC₅₀: 9 nM					99.57%
7-Deazaguanine	DYRK1A						99.73%
Dyrk1A-IN-4	DYRK1A, IC₅₀: 2 nM	DYRK2, IC₅₀: 6 nM					99.30%
MU1210		DYRK2, IC₅₀: 1309 nM					99.50%
EHT 5372	DYRK1A, IC₅₀: 0.22 nM DYRK1B, IC₅₀: 0.28 nM	DYRK2, IC₅₀: 10.8 nM		DYRK4, IC₅₀: 93.2 nM			98.12%
CLK1-IN-3	DYRK1A, IC₅₀: 1521 nM						98.54%
ON 108600	DYRK1A, IC₅₀: 0.016 μM DYRK1B, IC₅₀: 0.007 μM	DYRK2, IC₅₀: 0.028 μM					98.65%
LDN-192960	DYRK1	DYRK2					99.58%
GNF2133 hydrochloride	DYRK1A, IC₅₀: 0.0062 μM						99.86%
HTH-01-091				DYRK4, IC₅₀: 41.8 nM			99.81%
LDN-209929 dihydrochloride		DYRK2					98.33%
DYRKs-IN-1 hydrochloride	DYRK1A, IC₅₀: 5 nM DYRK1B, IC₅₀: 8 nM						98.29%
ZJCK-6-46	DYRK1A, IC₅₀: 0.68 nM DYRK1B, IC₅₀: 1.02 nM	DYRK2, IC₅₀: 14.18 nM	DYRK3, IC₅₀: 17.48 nM	DYRK4, IC₅₀: 401.3 nM			99.06%
KH-CB20	DYRK1A, IC₅₀: 57.8 nM						99.80%
LDN-192960 hydrochloride	DYRK1	DYRK2					99.76%
RD0392	DYRK1A						99.93%
DS12881479	DYRK1A						99.63%
Dyrk1A-IN-13	DYRK1A, IC₅₀: 41 nM DYRK1B, IC₅₀: 78 nM						99.43%
DYRKs-IN-1	DYRK1A, IC₅₀: 5 nM DYRK1B, IC₅₀: 8 nM
(R)-(+)-O-Demethylbuchenavianine	DYRK1A						98.67%
MBM-55S	DYRK1A, IC₅₀: 6.5 nM
Dyrk1A/B-IN-1	DYRK1A, Ki: 67.8 nM DYRK1B, Ki: 237.9 nM
Haspin-IN-2	DYRK1A, IC₅₀: 917 nM
Atalaphyllidine	DYRK1A, IC₅₀: 2.2 μM
VS-II-173	DYRK1
JH-XVII-10	DYRK1A, IC₅₀: 3 nM DYRK1B, IC₅₀: 5 nM
ARN25699	DYRK1A
GSK3-IN-10	DYRK1A, IC₅₀: 170 nM DYRK1B, IC₅₀: 47 nM	DYRK2, IC₅₀: 800 nM
Dyrk1A-IN-15	DYRK1A, IC₅₀: 19 nM
Dyrk1A/α-synuclein-IN-1	DYRK1A, IC₅₀: 177 nM
Dyrk1A-IN-7	DYRK1A, IC₅₀: 28 nM
Dyrk1A-IN-16	DYRK1A, IC₅₀: 50 nM
Dyrk1A-IN-1	DYRK1
DYRK2 ligand 1		DYRK2
XRF-1021					HIPK2, IC₅₀: 0.18 μM
UNC9750	DYRK1B
PROTAC DYRK2 degrader 1		DYRK2, DC₅₀: 1.607 μM
Dyrk1A/α-synuclein-IN-2	DYRK1A
hAChE-IN-8	DYRK1A, IC₅₀: >10 μM
MU1787	DYRK1A, IC₅₀: 213 nM DYRK1B, IC₅₀: 956 nM	DYRK2, IC₅₀: 1309 nM			HIPK1, IC₅₀: 285 nM HIPK2, IC₅₀: 123 nM HIPK3, IC₅₀: 283 nM
JH-XIV-68-3	DYRK1
KTD-092	DYRK1A, IC₅₀: 22 nM
Dyrk1A-IN-8	DYRK1A, IC₅₀: 209 nM
Haspin-IN-1	DYRK1A, IC₅₀: 916.3 nM
2-Methyl-5-acetylphenol					HIPK2
Dyrk1A-IN-17	DYRK1A
Cnksr3 Rat Pre-designed siRNA Set A						PRP4
Norharmine	DYRK1A
Dyrk1A-IN-11	DYRK1A, EC₅₀: 0.0021 μM
Hipk2 Rat Pre-designed siRNA Set A					HIPK1
RD0448	DYRK1A, IC₅₀: >64 μM DYRK1B, IC₅₀: 52 μM	DYRK2, IC₅₀: 31 μM
Dyrk1A-IN-2	DYRK1A, EC₅₀: 37 nM
Dyrk1A-IN-12	DYRK1A, IC₅₀: 95 nM

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