1. Signaling Pathways
  2. Protein Tyrosine Kinase/RTK
  3. DYRK
  4. DYRK Inhibitors

DYRK Inhibitors

DYRK1

DYRK2

DYRK4

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

DYRK Inhibitors
Product Name DYRK1 DYRK2 DYRK4 Purity
AZ191
DYRK1B
    99.98%
Dyrk1A-IN-7
DYRK1A, IC50: 28 nM
   
T025
DYRK1A, Kd: 0.074 nM
DYRK1B, Kd: 1.5 nM
DYRK2, Kd: 32 nM
  98.84%
DYRK1-IN-1
DYRK1A, IC50: 220 nM
DYRK1A, Kd: 3 nM
DYRK1B, Kd: 56 nM
    99.62%
GNF2133
DYRK1A, IC50: 0.0062 μM
    98.49%
Protein kinase inhibitor 1 hydrochloride
DYRK1
DYRK2
  ≥98.0%
ILK-IN-3
DYRK1
    99.62%
Harmine hydrochloride
DYRK1A
    99.93%
EHT 5372
DYRK1A, IC50: 0.22 nM
DYRK1B, IC50: 0.28 nM
DYRK2, IC50: 10.8 nM
DYRK4, IC50: 93.2 nM
98.12%
ML167
DYRK1A, IC50: >10000 nM
DYRK1B, IC50: 4420 nM
    98.62%
AZ-Dyrk1B-33
DYRK1B
    99.95%
Dyrk1A-IN-5
DYRK1A, IC50: 6 nM
DYRK1B, IC50: 600 nM
DYRK2, IC50: >10000 nM
  98.56%
KH-CB20
DYRK1A, IC50: 57.8 nM
    99.80%
GNF4877
DYRK1A, IC50: 6 nM
    99.32%
CLK1-IN-3
DYRK1A, IC50: 1521 nM
    98.03%
Dyrk1A-IN-4
DYRK1A, IC50: 2 nM
DYRK2, IC50: 6 nM
  99.90%
HTH-01-091    
DYRK4, IC50: 41.8 nM
98.64%
DYRKs-IN-1
DYRK1A, IC50: 5 nM
DYRK1B, IC50: 8 nM
   
DYRKs-IN-1 hydrochloride
DYRK1A, IC50: 5 nM
DYRK1B, IC50: 8 nM
    99.70%
MBM-55S
DYRK1A, IC50: 6.5 nM
   
Dyrk1A/B-IN-1
DYRK1A, Ki: 67.8 nM
DYRK1B, Ki: 237.9 nM
   
Haspin-IN-2
DYRK1A, IC50: 917 nM
   
JH-XVII-10
DYRK1A, IC50: 3 nM
DYRK1B, IC50: 5 nM
   
Dyrk1A/α-synuclein-IN-1
DYRK1A, IC50: 177 nM
   
Dyrk1A-IN-1
DYRK1
   
ON 108600
DYRK1A, IC50: 0.016 μM
DYRK1B, IC50: 0.007 μM
DYRK2, IC50: 0.028 μM
  99.73%
Dyrk1A/α-synuclein-IN-2
DYRK1A
   
JH-XIV-68-3
DYRK1
   
Haspin-IN-1
DYRK1A, IC50: 916.3 nM
   
GNF2133 hydrochloride
DYRK1A, IC50: 0.0062 μM
   
Dyrk1A-IN-2
DYRK1A, EC50: 37 nM