PCSK9 - proprotein convertase subtilisin/kexin type 9 Gene
Species: Sus scrofa
Gene Type: protein coding
Gene ID: 100620501
PCSK9 Products (1)
| mRNA | Protein | Name |
|---|---|---|
| XM_005653438.3 | XP_005653495.2 | LOW QUALITY PROTEIN: proprotein convertase subtilisin/kexin type 9 |
| Protein Preferred Names | Protein Names | |
|---|---|---|
|
LOW QUALITY PROTEIN: proprotein convertase subtilisin/kexin type 9 |
|
Related Agents
- Approval
- Clinical Phase
- Pre-clinical Phase
Approval
Bioactive Molecules
(3)
| Cat. No. | Product Name |
Effect
|
Purity |
Rare Diseases
|
|---|---|---|---|---|
| HY-132591A | Inclisiran sodium | Inhibitor | 99.08% | Unkown |
| HY-132591 | Inclisiran | Inhibitor | 99.48% | Unkown |
| HY-132591C | Inclisiran sodium scrambled negative control | Inhibitor | / | Unkown |
Bioactive MoleculesInhibitory Antibodies
(2)
| Cat. No. | Product Name |
Effect
|
Purity |
Rare Diseases
|
|---|---|---|---|---|
| HY-P9928 | Alirocumab | Inhibitor | 97.00% | Unkown |
| HY-P99696 | Lerodalcibep | / | Unkown |
Clinical Phase
Bioactive Molecules
(4)
| Cat. No. | Product Name |
Effect
|
Purity |
Phase |
|---|---|---|---|---|
| HY-12090 | Anacetrapib | Inhibitor | 99.25% | Phase 3 |
| HY-158825 | Cepadacursen sodium | / | Phase 2 | |
| HY-148687A | SPC5001 sodium | Inhibitor | 98.89% | Phase 1 |
| HY-112598 | PF-06815345 | Inhibitor | / | Phase 1 |
Bioactive MoleculesInhibitory Antibodies
(6)
| Cat. No. | Product Name |
Effect
|
Purity |
Phase |
|---|---|---|---|---|
| HY-P99822 | Recaticimab | Inhibitor | 99.71% | Phase 4 |
| HY-P99552 | Tafolecimab | Inhibitor | 95.04% | Phase 4 |
| HY-P99187 | Bococizumab | Inhibitor | 99.80% | Phase 3 |
| HY-P99871 | Ebronucimab | Inhibitor | / | Phase 3 |
| HY-P99773 | Ongericimab | Inhibitor | / | Phase 3 |
| HY-P99626 | Frovocimab | Inhibitor | 96.78% | Phase 2 |
Pre-clinical Phase
Bioactive Molecules
(72)
| Cat. No. | Product Name |
Effect
|
Purity |
Rare Diseases
|
|---|---|---|---|---|
| HY-148673 | Laroprovstat | Inhibitor | 99.93% | Unkown |
| HY-P4153 | Enlicitide chloride | Inhibitor | 99.63% | Unkown |
| HY-120088A | PF-06446846 hydrochloride | Inhibitor | 99.44% | Unkown |
| HY-143219 | SS-Inclisiran sodium | Inhibitor | 97.91% | Unkown |
| HY-12402 | SBC-115076 | Inhibitor | 99.28% | Unkown |
| HY-P2276 | Pep2-8 | Inhibitor | 99.74% | Unkown |
| HY-W510159 | 5-O-Methylembelin | Inhibitor | 99.43% | Unkown |
| HY-143220 | SS(no Galnac)-Inclisiran sodium | Inhibitor | 98.05% | Unkown |
| HY-150223 | GalNAc unconjugated/naked Inclisiran | Inhibitor | 94.67% | Unkown |
| HY-152221 | PCSK9-IN-10 | Inhibitor | 98.89% | Unkown |
| HY-152223 | PCSK9-IN-11 | Inhibitor | 99.30% | Unkown |
| HY-101354 | R-IMPP | Inhibitor | 99.93% | Unkown |
| HY-157434 | PCSK9-IN-23 | Inhibitor | 99.57% | Unkown |
| HY-148758 | PCSK9-IN-13 | Inhibitor | 98.00% | Unkown |
| HY-130245 | PCSK9 degrader 1 | Degrader | 98.33% | Unkown |
| HY-101832 | SBC-110736 | Inhibitor | 99.55% | Unkown |
| HY-141714 | SBC-115337 | Inhibitor | 98.02% | Unkown |
| HY-163794 | DC371739 | Inhibitor | 95.56% | Unkown |
| HY-158827A | AZD8233 sodium | 94.99% | Unkown | |
| HY-120088 | PF-06446846 | Inhibitor | 98.35% | Unkown |
| HY-142026 | Vitisin A | Inhibitor | 96% | Unkown |
| HY-162562 | E28362 | Inhibitor | 94.51% | Unkown |
| HY-161939 | 7030B-C5 | Inhibitor | 99.78% | Unkown |
| HY-P2276A | Pep2-8 TFA | Inhibitor | 98.78% | Unkown |
| HY-161940 | PCSK9-IN-30 | Inhibitor | / | Unkown |
| HY-148687 | SPC5001 | Inhibitor | 95.11% | Unkown |
| HY-147252A | Bezeparsen sodium | Inhibitor | 95.21% | Unkown |
| HY-112598A | PF-06815345 hydrochloride | Inhibitor | 98.15% | Unkown |
| HY-159595 | PCSK9-IN-29 | Inhibitor | 99.44% | Unkown |
| HY-148626 | CVI-LM001 | Inhibitor | / | Unkown |
| HY-W1126955 | Enlicitide (decanoate) | Inhibitor | / | Unkown |
| HY-147252 | Bezeparsen | Inhibitor | / | Unkown |
| HY-148689 | SPC4061 | Inhibitor | / | Unkown |
| HY-RS10177 | PCSK9 Human Pre-designed siRNA Set A | Inhibitor | / | Unkown |
| HY-149310 | Dim16 | Inhibitor | / | Unkown |
| HY-161435 | PCSK9-IN-27 | Inhibitor | / | Unkown |
| HY-153453 | PCSK9-IN-17 | Inhibitor | / | Unkown |
| HY-179106 | PCSK9-IN-34 | Inhibitor | / | Unkown |
| HY-161434 | PCSK9-IN-26 | Inhibitor | / | Unkown |
| HY-P11071 | PCSK9 Inhibitor, EGF-A | Inhibitor | / | Unkown |
| HY-153452 | PCSK9-IN-16 | Inhibitor | / | Unkown |
| HY-130245A | (R,R)-PCSK9 degrader 1 | Degrader | / | Unkown |
| HY-N10702 | PCSK9-IN-9 | Inhibitor | / | Unkown |
| HY-134482 | PCSK9-IN-1 | Inhibitor | / | Unkown |
| HY-148687C | SPC5001 sodium scrambled negative control | Inhibitor | / | Unkown |
| HY-141724 | PCSK9 ligand 1 | Inhibitor | / | Unkown |
| HY-163141 | PCSK9-IN-24 | Inhibitor | / | Unkown |
| HY-153454 | PCSK9-IN-18 | Inhibitor | / | Unkown |
| HY-P11216 | Pep2-8 analogue 18 | Inhibitor | / | Unkown |
| HY-153391 | PCSK9-IN-14 | Inhibitor | / | Unkown |
| HY-160036 | PCSK9-IN-22 | Inhibitor | / | Unkown |
| HY-146085 | PCSK9 modulator-4 | Modulator | / | Unkown |
| HY-128334 | PCSK9 modulator-2 | Modulator | / | Unkown |
| HY-148689C | SPC4061 sodium scrambled negative control | Inhibitor | / | Unkown |
| HY-176043 | PCSK9 autophagic degrader 2 | Degrader | / | Unkown |
| HY-146084 | PCSK9 modulator-3 | Modulator | / | Unkown |
| HY-161942 | PCSK9-IN-31 | Inhibitor | / | Unkown |
| HY-153451 | PCSK9-IN-15 | Inhibitor | / | Unkown |
| HY-148689A | SPC4061 sodium | Inhibitor | / | Unkown |
| HY-161941 | MeIm | Inhibitor | / | Unkown |
| HY-155006 | PCSK9-IN-19 | Inhibitor | / | Unkown |
| HY-147252C | Bezeparsen sodium scrambled negative control | Inhibitor | / | Unkown |
| HY-164344 | PCSK9 allosteric binder-1 | / | Unkown | |
| HY-168156 | PCSK9-IN-32 | Inhibitor | / | Unkown |
| HY-18778C | Obicetrapib hemicalcium | Inhibitor | / | Unkown |
| HY-158825A | Cepadacursen sodium scrambled negative control | / | Unkown | |
| HY-175189 | PCSK9-IN-33 | Inhibitor | / | Unkown |
| HY-161938 | BRD8518 | Inhibitor | / | Unkown |
| HY-158827 | AZD8233 | / | Unkown | |
| HY-158827B | AZD8233 sodium scrambled negative control | / | Unkown | |
| HY-155415 | PCSK9-IN-20 | Inhibitor | / | Unkown |
| HY-149310A | Dim16 hydrochloride | Inhibitor | / | Unkown |
Bioactive MoleculesInhibitory Antibodies
(8)
| Cat. No. | Product Name |
Effect
|
Purity |
Rare Diseases
|
|---|---|---|---|---|
| HY-P9928A | Alirocumab (anti-PCSK9) | Inhibitor | 98.24% | Unkown |
| HY-P99816 | Ralpancizumab | Inhibitor | 96.23% | Unkown |
| HY-P99251 | Lodelcizumab | Inhibitor | ≥99.0% | Unkown |
| HY-P99251 | Lodelcizumab | Inhibitor | ≥99.0% | Unkown |
| HY-P991721 | Ticalicibart | Inhibitor | 99.028% | Unkown |
| HY-P992407 | MEDI-4166 | / | Unkown | |
| HY-P991343 | ALD306 | Inhibitor | / | Unkown |
| HY-P990485 | Anti-PCSK9 Antibody | Inhibitor | 98.39% | Unkown |