1. GPCR/G Protein Neuronal Signaling
  2. Melanocortin Receptor
  3. hMC1R agonist 1

(EC50=3 nM). hMC1R agonist 1 shows at least 300-fold selectivity for hMC1R over hMC3R (b>EC50=902 nM), hMC4R (b>EC50=915 nM), and hMC5R (b>EC50=>1000 nM). hMC1R agonist 1 has the potential for the therapeutic intervention of melanocortin family.

For research use only. We do not sell to patients.

hMC1R agonist 1 Chemical Structure

hMC1R agonist 1 Chemical Structure

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Description

(EC50=3 nM). hMC1R agonist 1 shows at least 300-fold selectivity for hMC1R over hMC3R (b>EC50=902 nM), hMC4R (b>EC50=915 nM), and hMC5R (b>EC50=>1000 nM). hMC1R agonist 1 has the potential for the therapeutic intervention of melanocortin family[1].

IC50 & Target

MC1R

 

Molecular Weight

1107.35

Formula

C54H70N14O8S2

SMILES

O=C([C@@H](NC(C)=O)CCCC)N[C@H](C(N[C@H](C(N[C@@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N)=O)CSC1)=O)CC2=CNC3=C2C=CC=C3)=O)CCCNC(N)=N)=O)CC4=CC=CC=C4)=O)CC5=CNC=N5)=O)CSCC6=CC1=CC=C6

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation
References
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hMC1R agonist 1 Related Classifications

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Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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hMC1R agonist 1
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HY-P99004
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