hMCH-1R antagonist 1
hMCH-1R antagonist 1 (Compound 30) is an effective and selective antagonist of human melanin-concentrating hormone receptor 1 (hMCHR1) with an KB value of 3.6 nM. HMCH-1R antagonist 1 can bind to hMCHR1 and hMCHR2 with IC50 values of 65 nM and 49 nM, respectively. HMCH-1R antagonistist 1 can be used for metabolic research.
For research use only. We do not sell to patients.
- CAS No.: 353487-64-6
- Formula: C49H82N16O11S3
- Molecular Weight:1167.47
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
Chemical Information
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CAS No. 353487-64-6
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Molecular Weight 1167.47
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Formula C49H82N16O11S3
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Sequence
Ac-Arg-Cys-Met-{5-Ava}-Arg-Val-Tyr-{5-Ava}-Cys-NH2 (Disulfide bridge: Cys2-Cys9)
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Sequence Shortening
Ac-RCM-{5-Ava}-RVY-{5-Ava}-C-NH2 (Disulfide bridge: Cys2-Cys9)
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
hMCH-1R antagonist 1 Related Classifications
HY-P4745 Related Classifications
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