2. GPCR/G Protein Neuronal Signaling Immunology/Inflammation
  3. Histamine Receptor
  4. Orf 17910

ORF 17910 is a potent, long-acting, orally active histamine H2 receptor antagonist. ORF 17910 exhibits significant and prolonged acid-suppressing activity in dogs and rats. However, the cardiac depressant effect of ORF 17910 cannot be completely overcome at high concentrations. ORF 17910 may be used to study diseases such as gastric ulcers.

For research use only. We do not sell to patients.

Orf 17910

Orf 17910 Chemical Structure

CAS No. : 87107-94-6

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Orf 17910 Related Antibodies

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Description

ORF 17910 is a potent, long-acting, orally active histamine H2 receptor antagonist. ORF 17910 exhibits significant and prolonged acid-suppressing activity in dogs and rats. However, the cardiac depressant effect of ORF 17910 cannot be completely overcome at high concentrations. ORF 17910 may be used to study diseases such as gastric ulcers[1].

IC50 & Target[1]

H2 Receptor

 

Molecular Weight

377.51

Formula

C18H27N5O2S
CAS No.
SMILES

O=S1N=C(N)C(=N1)NCCCOC2=CC=CC(=C2)CN3CCC(C)CC3
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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Orf 17910 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Orf 1791087107-94-6Orf17910Orf-17910Histamine ReceptorInhibitorinhibitorinhibit

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