1. GPCR/G Protein Neuronal Signaling
  2. Dopamine Receptor
  3. Raxlaprazine etomoxil

Raxlaprazine etomoxil is a small molecule compound with dopamine D2 and D3 receptor modulating activity, which has potential application value in research related to mental illnesses. Raxlaprazine etomoxil exhibits high affinity for human recombinant D2L receptors, with an inhibition constant (Ki) of 1.95 nM. Raxlaprazine etomoxil effectively inhibits forskolin-stimulated cAMP accumulation, with an half maximal effective concentration (EC50) of 3.72 nM in functional activity experiments.

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Raxlaprazine etomoxil

Raxlaprazine etomoxil Chemische Struktur

CAS. Nr. : 3034857-88-7

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Beschreibung

Raxlaprazine etomoxil is a small molecule compound with dopamine D2 and D3 receptor modulating activity, which has potential application value in research related to mental illnesses. Raxlaprazine etomoxil exhibits high affinity for human recombinant D2L receptors, with an inhibition constant (Ki) of 1.95 nM. Raxlaprazine etomoxil effectively inhibits forskolin-stimulated cAMP accumulation, with an half maximal effective concentration (EC50) of 3.72 nM in functional activity experiments[1].

Molekulargewicht

471.46

Formel

C23H36Cl2N4O2

CAS. Nr.
SMILES

ClC1=C(C=CC=C1Cl)N2CCN(CC2)CC[C@H]3CC[C@@H](CC3)NC(N(C)COCC)=O

Versand

Room temperature in continental US; may vary elsewhere.

Speicherung

Please store the product under the recommended conditions in the Certificate of Analysis.

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Raxlaprazine etomoxil
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