2. (S)-Remoxipride hydrochloride

(S)-Remoxipride hydrochloride  (Synonyms: (-)-Remoxipride hydrochloride)

Cat. No.: HY-101313A Purity: 99.93%
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(S)-Remoxipride ((-)-Remoxipride) hydrochloride is a selective dopamine D2-receptor antagonist with an IC50 value of 1.57 μM. (S)-Remoxipride hydrochloride can be used for the research of psychotic disorder.

For research use only. We do not sell to patients.

(S)-Remoxipride hydrochloride Chemical Structure

(S)-Remoxipride hydrochloride Chemical Structure

CAS No. : 73220-03-8

Size Price Stock Quantity
5 mg USD 110 In-stock
10 mg USD 170 In-stock
25 mg USD 340 In-stock
50 mg USD 510 In-stock
100 mg USD 750 In-stock
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Other Forms of (S)-Remoxipride hydrochloride:

(S)-Remoxipride hydrochloride Related Antibodies

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Description

(S)-Remoxipride ((-)-Remoxipride) hydrochloride is a selective dopamine D2-receptor antagonist with an IC50 value of 1.57 μM. (S)-Remoxipride hydrochloride can be used for the research of psychotic disorder[1].
In Vitro

(S)-Remoxipride hydrochloride (1-100 μM; 20 min) shows binding efficiency with IC50s of ＞100, 1.57 and 42 μM for dopamine D1, dopamine D2 and α1-Adrenoccptor, respectively[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

(S)-Remoxipride hydrochloride Related Antibodies
In Vivo

(S)-Remoxipride hydrochloride (0.1-100 μM/kg; i.p. 60 min prior to apomorphine) blockades apomorphine-induced behaviors s in rats and vomiting in dogs[1].
(S)-Remoxipride hydrochloride (0.1-10 mg/kg; i.p. 30 min prior to apomorphine) displaces [3H]spiperone from both striatal and extra-striatal areas[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Molecular Weight

407.73

Formula

C16H24BrClN2O3
CAS No.
Appearance

Solid

Color

White to off-white

SMILES

O=C(NC[C@H]1N(CC)CCC1)C2=C(OC)C=CC(Br)=C2OC.Cl
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

4°C, sealed storage, away from moisture

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

Solvent & Solubility
In Vitro: 

DMSO : 62.5 mg/mL (153.29 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.4526 mL 12.2630 mL 24.5260 mL
5 mM 0.4905 mL 2.4526 mL 4.9052 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

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Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass
=
Concentration
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Volume
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Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start)

C1

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Volume (start)

V1

=
Concentration (final)

C2

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V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

Dosage

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g

Dosing volume
(per animal)

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Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
Purity & Documentation

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 2.4526 mL 12.2630 mL 24.5260 mL 61.3151 mL
5 mM 0.4905 mL 2.4526 mL 4.9052 mL 12.2630 mL
10 mM 0.2453 mL 1.2263 mL 2.4526 mL 6.1315 mL
15 mM 0.1635 mL 0.8175 mL 1.6351 mL 4.0877 mL
20 mM 0.1226 mL 0.6132 mL 1.2263 mL 3.0658 mL
25 mM 0.0981 mL 0.4905 mL 0.9810 mL 2.4526 mL
30 mM 0.0818 mL 0.4088 mL 0.8175 mL 2.0438 mL
40 mM 0.0613 mL 0.3066 mL 0.6132 mL 1.5329 mL
50 mM 0.0491 mL 0.2453 mL 0.4905 mL 1.2263 mL
60 mM 0.0409 mL 0.2044 mL 0.4088 mL 1.0219 mL
80 mM 0.0307 mL 0.1533 mL 0.3066 mL 0.7664 mL
100 mM 0.0245 mL 0.1226 mL 0.2453 mL 0.6132 mL
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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

(S)-Remoxipride73220-03-8(-)-RemoxiprideInhibitorinhibitorinhibit

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