(S)-Remoxipride hydrochloride
Based on 1 Customer Validation
(S)-Remoxipride ((-)-Remoxipride) hydrochloride is a selective dopamine D2-receptor antagonist with an IC50 value of 1.57 μM. (S)-Remoxipride hydrochloride can be used for the research of psychotic disorder.
For research use only. We do not sell to patients.
- Purity: 99.75%
- CAS No.: 73220-03-8
- Formula: C16H24BrClN2O3
- Molecular Weight:407.73
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Storage:
4°C, sealed storage, away from moisture
* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
All Dopamine Receptor Isoforms
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Biological Activity
(S)-Remoxipride hydrochloride (1-100 μM; 20 min) shows binding efficiency with IC50s of >100, 1.57 and 42 μM for dopamine D1, dopamine D2 and α1-Adrenoccptor, respectively[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 73220-03-8
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Appearance Solid
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Molecular Weight 407.73
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Formula C16H24BrClN2O3
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Color White to off-white
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SMILES
O=C(NC[C@H]1N(CC)CCC1)C2=C(OC)C=CC(Br)=C2OC.Cl
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Synonyms
(-)-Remoxipride hydrochloride
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
4°C, sealed storage, away from moisture
* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
Solvent & Solubility
H2O : 100 mg/mL (245.26 mM; Need ultrasonic)
DMSO : 62.5 mg/mL (153.29 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
* Note: If you choose water as the stock solution, please dilute it to the working solution, then filter and sterilize it with a 0.22 μm filter before use.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
* Note: If you choose water as the stock solution, please dilute it to the working solution, then filter and sterilize it with a 0.22 μm filter before use.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Purity & Documentation
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Data Sheet (274 KB)
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SDS (252 KB)
- English - EN (252 KB)
- Français - FR (252 KB)
- Deutsch - DE (252 KB)
- Norwegian - NO (252 KB)
- Español - ES (252 KB)
- Swedish - SV (252 KB)
- Italian - IT (252 KB)
- Korean - KR (252 KB)
- Portuguese - PT (252 KB)
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Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO / H2O | 1 mM | 2.4526 mL | 12.2630 mL | 24.5260 mL | 61.3151 mL |
| 5 mM | 0.4905 mL | 2.4526 mL | 4.9052 mL | 12.2630 mL | |
| 10 mM | 0.2453 mL | 1.2263 mL | 2.4526 mL | 6.1315 mL | |
| 15 mM | 0.1635 mL | 0.8175 mL | 1.6351 mL | 4.0877 mL | |
| 20 mM | 0.1226 mL | 0.6132 mL | 1.2263 mL | 3.0658 mL | |
| 25 mM | 0.0981 mL | 0.4905 mL | 0.9810 mL | 2.4526 mL | |
| 30 mM | 0.0818 mL | 0.4088 mL | 0.8175 mL | 2.0438 mL | |
| 40 mM | 0.0613 mL | 0.3066 mL | 0.6132 mL | 1.5329 mL | |
| 50 mM | 0.0491 mL | 0.2453 mL | 0.4905 mL | 1.2263 mL | |
| 60 mM | 0.0409 mL | 0.2044 mL | 0.4088 mL | 1.0219 mL | |
| 80 mM | 0.0307 mL | 0.1533 mL | 0.3066 mL | 0.7664 mL | |
| 100 mM | 0.0245 mL | 0.1226 mL | 0.2453 mL | 0.6132 mL |
* Note: If you choose water as the stock solution, please dilute it to the working solution, then filter and sterilize it with a 0.22 μm filter before use.